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Target
Nociceptin receptor
Ligand
BDBM50475328
Substrate
n/a
Meas. Tech.
ChEMBL_313609 (CHEMBL835016)
EC50
0.436516±n/a nM
Citation
 Guerrini, R; Caló, G; Lambert, DG; Carrá, G; Arduin, M; Barnes, TA; McDonald, J; Rizzi, D; Trapella, C; Marzola, E; Rowbotham, DJ; Regoli, D; Salvadori, S N- and C-terminal modifications of nociceptin/orphanin FQ generate highly potent NOP receptor ligands. J Med Chem 48:1421-7 (2005) [PubMed]  Article 
Target
Name:
Nociceptin receptor
Synonyms:
Orphanin FQ receptor | KOR-3 | Kappa-type 3 opioid receptor | K3 opiate receptor | ORGC | Nociceptin receptor | OPRX_MOUSE | Oprl1 | Oor | Oprl | Nociceptin/Orphanin FQ, NOP receptor
Type:
Enzyme Catalytic Domain
Mol. Mass.:
40499.09
Organism:
Mouse
Description:
Nociceptin/Orphanin FQ, NOP receptor 0 MOUSE::P35377
Residue:
367
Sequence:
MESLFPAPFWEVLYGSHFQGNLSLLNETVPHHLLLNASHSAFLPLGLKVTIVGLYLAVCIGGLLGNCLVMYVILRHTKMKTATNIYIFNLALADTLVLLTLPFQGTDILLGFWPFGNALCKTVIAIDYYNMFTSTFTLTAMSVDRYVAICHPIRALDVRTSSKAQAVNVAIWALASVVGVPVAIMGSAQVEDEEIECLVEIPAPQDYWGPVFAICIFLFSFIIPVLIISVCYSLMIRRLRGVRLLSGSREKDRNLRRITRLVLVVVAVFVGCWTPVQVFVLVQGLGVQPGSETAVAILRFCTALGYVNSCLNPILYAFLDENFKACFRKFCCASALHREMQVSDRVRSIAKDVGLGCKTSETVPRPA
  
Inhibitor
Name:
BDBM50475328
Synonyms:
CHEMBL414782
Type:
Small organic molecule
Emp. Form.:
TBD
Mol. Mass.:
TBD
SMILES:
TBD
Structure:
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