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Target
Mu-type opioid receptor
Ligand
BDBM50370595
Substrate
n/a
Meas. Tech.
ChEMBL_978254 (CHEMBL2423623)
EC50
160±n/a nM
Citation
 Magnus, P; Ghavimi, B; Coe, JW Access to 7β-analogs of codeine with mixed μ/δ agonist activity via 6,7-α-epoxide opening. Bioorg Med Chem Lett 23:4870-4 (2013) [PubMed]  Article 
Target
Name:
Mu-type opioid receptor
Synonyms:
OPIATE Mu | M-OR-1 | MOR-1 | OPRM_MOUSE | Oprm1 | Mor | Oprm | Opioid receptors; mu and delta
Type:
Enzyme Catalytic Domain
Mol. Mass.:
44431.62
Organism:
Mouse
Description:
OPIATE Mu OPRM1 MOUSE::P42866
Residue:
398
Sequence:
MDSSAGPGNISDCSDPLAPASCSPAPGSWLNLSHVDGNQSDPCGPNRTGLGGSHSLCPQTGSPSMVTAITIMALYSIVCVVGLFGNFLVMYVIVRYTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGNILCKIVISIDYYNMFTSIFTLCTMSVDRYIAVCHPVKALDFRTPRNAKIVNVCNWILSSAIGLPVMFMATTKYRQGSIDCTLTFSHPTWYWENLLKICVFIFAFIMPVLIITVCYGLMILRLKSVRMLSGSKEKDRNLRRITRMVLVVVAVFIVCWTPIHIYVIIKALITIPETTFQTVSWHFCIALGYTNSCLNPVLYAFLDENFKRCFREFCIPTSSTIEQQNSARIRQNTREHPSTANTVDRTNHQLENLEAETAPLP
  
Inhibitor
Name:
BDBM50370595
Synonyms:
US9233167, Oxycodone | Oxycontin | OXYCODONE | US1184575, oxycodone
Type:
Small organic molecule
Emp. Form.:
TBD
Mol. Mass.:
TBD
SMILES:
TBD
Structure:
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