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Target
P2Y purinoceptor 4
Ligand
BDBM50496855
Substrate
n/a
Meas. Tech.
ChEMBL_1330931 (CHEMBL3224911)
EC50
7440±n/a nM
Citation
 Jayasekara, PS; Barrett, MO; Ball, CB; Brown, KA; Kozma, E; Costanzi, S; Squarcialupi, L; Balasubramanian, R; Maruoka, H; Jacobson, KA 4-Alkyloxyimino-cytosine nucleotides: tethering approaches to molecular probes for the P2Y Medchemcomm 4:1156-1165 (2013) [PubMed]  Article 
Target
Name:
P2Y purinoceptor 4
Synonyms:
P2P | P2Y purinoceptor 4 | P2Y4 | UNR | Uridine nucleotide receptor | P2RY4_HUMAN | P2RY4 | NRU | Pyrimidinergic receptor P2Y4
Type:
PROTEIN
Mol. Mass.:
40977.17
Organism:
Human
Description:
ChEMBL_751027
Residue:
365
Sequence:
MASTESSLLRSLGLSPGPGSSEVELDCWFDEDFKFILLPVSYAVVFVLGLGLNAPTLWLFIFRLRPWDATATYMFHLALSDTLYVLSLPTLIYYYAAHNHWPFGTEICKFVRFLFYWNLYCSVLFLTCISVHRYLGICHPLRALRWGRPRLAGLLCLAVWLVVAGCLVPNLFFVTTSNKGTTVLCHDTTRPEEFDHYVHFSSAVMGLLFGVPCLVTLVCYGLMARRLYQPLPGSAQSSSRLRSLRTIAVVLTVFAVCFVPFHITRTIYYLARLLEADCRVLNIVNVVYKVTRPLASANSCLDPVLYLLTGDKYRRQLRQLCGGGKPQPRTAASSLALVSLPEDSSCRWAATPQDSSCSTPRADRL
  
Inhibitor
Name:
BDBM50496855
Synonyms:
CHEMBL3220048
Type:
Small organic molecule
Emp. Form.:
C16H20BrN3O12P2
Mol. Mass.:
588.2
SMILES:
O[C@@H]1[C@@H](COP(O)(=O)OP(O)(O)=O)O[C@H]([C@@H]1O)n1cc\c(=N\OCc2ccc(Br)cc2)[nH]c1=O |r|
Structure:
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