Target
Myeloblastin
Ligand
BDBM50502660
Substrate
n/a
Meas. Tech.
ChEMBL_1808142 (CHEMBL4307501)
Ki
245±n/a nM
Citation
 Tian, SSwedberg, JELi, CYCraik, DJde Veer, SJ Iterative Optimization of the Cyclic Peptide SFTI-1 Yields Potent Inhibitors of Neutrophil Proteinase 3. ACS Med Chem Lett 10:1234-1239 (2019) [PubMed]  Article 
Target
Name:
Myeloblastin
Synonyms:
PRTN3_HUMAN | PRTN3 | MBN | Leukocyte proteinase 3
Type:
PROTEIN
Mol. Mass.:
27816.30
Organism:
Human
Description:
ChEMBL_1463425
Residue:
256
Sequence:
MAHRPPSPALASVLLALLLSGAARAAEIVGGHEAQPHSRPYMASLQMRGNPGSHFCGGTLIHPSFVLTAAHCLRDIPQRLVNVVLGAHNVRTQEPTQQHFSVAQVFLNNYDAENKLNDVLLIQLSSPANLSASVATVQLPQQDQPVPHGTQCLAMGWGRVGAHDPPAQVLQELNVTVVTFFCRPHNICTFVPRRKAGICFGDSGGPLICDGIIQGIDSFVIWGCATRLFPDFFTRVALYVDWIRSTLRRVEAKGRP
  
Inhibitor
Name:
BDBM50502660
Synonyms:
CHEMBL4469546
Type:
Small organic molecule
Emp. Form.:
TBD
Mol. Mass.:
TBD
SMILES:
TBD
Structure:
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