Reaction Details Report a problem with these data
Target
Myosin light chain kinase family member 4
Ligand
BDBM50505859
Substrate
n/a
Meas. Tech.
ChEMBL_1824429 (CHEMBL4324193)
IC50
10000±n/a nM
Citation
Röhm, S; Berger, BT; Schröder, M; Chaikuad, A; Winkel, R; Hekking, KFW; Benningshof, JJC; Müller, G; Tesch, R; Kudolo, M; Forster, M; Laufer, S; Knapp, S Fast Iterative Synthetic Approach toward Identification of Novel Highly Selective p38 MAP Kinase Inhibitors. J Med Chem 62:10757-10782 (2019) [PubMed] Article
More Info.:
Target
Name:
Myosin light chain kinase family member 4
Synonyms:
MYLK4 | MYLK4_HUMAN | SGK085
Type:
PROTEIN
Mol. Mass.:
44505.40
Organism:
Homo sapiens (Human)
Description:
ChEMBL_774289
Residue:
388
Sequence:
MLKVKRLEEFNTCYNSNQLEKMAFFQCREEVEKVKCFLEKNSGDQDSRSGHNEAKEVWSNADLTERMPVKSKRTSALAVDIPAPPAPFDHRIVTAKQGAVNSFYTVSKTEILGGGRFGQVHKCEETATGLKLAAKIIKTRGMKDKEEVKNEISVMNQLDHANLIQLYDAFESKNDIVLVMEYVDGGELFDRIIDESYNLTELDTILFMKQICEGIRHMHQMYILHLDLKPENILCVNRDAKQIKIIDFGLARRYKPREKLKVNFGTPEFLAPEVVNYDFVSFPTDMWSVGVIAYMLLSGLSPFLGDNDAETLNNILACRWDLEDEEFQDISEEAKEFISKLLIKEKSWRISASEALKHPWLSDHKLHSRLNAQKKKNRGSDAQDFVTK