Reaction Details Report a problem with these data
Target
Neurotensin receptor type 2
Ligand
BDBM50509510
Substrate
n/a
Meas. Tech.
ChEMBL_1838608 (CHEMBL4338741)
Ki
1.2±n/a nM
Citation
 Keller, M; Mahuroof, SA; Hong Yee, V; Carpenter, J; Schindler, L; Littmann, T; Pegoli, A; Hübner, H; Bernhardt, G; Gmeiner, P; Holliday, ND Fluorescence Labeling of Neurotensin(8-13) via Arginine Residues Gives Molecular Tools with High Receptor Affinity. ACS Med Chem Lett 11:16-22 (2020) [PubMed]  Article 
Target
Name:
Neurotensin receptor type 2
Synonyms:
Neurotensin receptor 2 | Levocabastine-sensitive neurotensin receptor | Neurotensin receptor type 2 | NTR2 receptor | NT-R-2 | NTR2 | NTR2_HUMAN | NTSR2 | Neurotensin receptor
Type:
PROTEIN
Mol. Mass.:
45404.76
Organism:
Human
Description:
ChEMBL_1281495
Residue:
410
Sequence:
METSSPRPPRPSSNPGLSLDARLGVDTRLWAKVLFTALYALIWALGAAGNALSAHVVLKARAGRAGRLRHHVLSLALAGLLLLLVGVPVELYSFVWFHYPWVFGDLGCRGYYFVHELCAYATVLSVAGLSAERCLAVCQPLRARSLLTPRRTRWLVALSWAASLGLALPMAVIMGQKHELETADGEPEPASRVCTVLVSRTALQVFIQVNVLVSFVLPLALTAFLNGVTVSHLLALCSQVPSTSTPGSSTPSRLELLSEEGLLSFIVWKKTFIQGGQVSLVRHKDVRRIRSLQRSVQVLRAIVVMYVICWLPYHARRLMYCYVPDDAWTDPLYNFYHYFYMVTNTLFYVSSAVTPLLYNAVSSSFRKLFLEAVSSLCGEHHPMKRLPPKPQSPTLMDTASGFGDPPETRT
  
Inhibitor
Name:
BDBM50509510
Synonyms:
CHEMBL4564746
Type:
Small organic molecule
Emp. Form.:
TBD
Mol. Mass.:
TBD
SMILES:
TBD
Structure:
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