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Target
Prostaglandin E synthase
Ligand
BDBM50569444
Substrate
n/a
Meas. Tech.
ChEMBL_2109352 (CHEMBL4818027)
IC50
340±n/a nM
Citation
 Kim, M; Kim, G; Kang, M; Ko, D; Nam, Y; Moon, CS; Kang, HM; Shin, JS; Werz, O; Lee, KT; Lee, JY Discovery of N-amido-phenylsulfonamide derivatives as novel microsomal prostaglandin E Bioorg Med Chem Lett 41:0 (2021) [PubMed]  Article 
Target
Name:
Prostaglandin E synthase
Synonyms:
Microsomal prostaglandin E synthase 1 | Prostaglandin E synthase | mPGES-1 | 5.3.99.3 | PTGES_MOUSE | Ptges | Pges
Type:
PROTEIN
Mol. Mass.:
17293.88
Organism:
Mouse
Description:
ChEMBL_104562
Residue:
153
Sequence:
MPSPGLVMESGQVLPAFLLCSTLLVIKMYAVAVITGQMRLRKKAFANPEDALKRGGLQYYRSDPDVERCLRAHRNDMETIYPFLFLGFVYSFLGPNPLIAWIHFLVVLTGRVVHTVAYLGKLNPRLRSGAYVLAQFSCFSMALQILWEVAHHL
  
Inhibitor
Name:
BDBM50569444
Synonyms:
CHEMBL4848472
Type:
Small organic molecule
Emp. Form.:
TBD
Mol. Mass.:
TBD
SMILES:
TBD
Structure:
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