Reaction Details Report a problem with these data
Target
Fibroblast growth factor 2
Ligand
BDBM50577061
Substrate
n/a
Meas. Tech.
ChEMBL_2129136 (CHEMBL4838565)
Kd
30000±n/a nM
Citation
Castelli, R; Taranto, S; Furiassi, L; Bozza, N; Marseglia, G; Ferlenghi, F; Rivara, S; Retini, M; Bedini, A; Spadoni, G; Matarazzo, S; Ronca, R; Presta, M; Mor, M; Giacomini, A Chemical modification of NSC12 leads to a specific FGF-trap with antitumor activity in multiple myeloma. Eur J Med Chem 221:0 (2021) [PubMed] Article
More Info.:
Target
Name:
Fibroblast growth factor 2
Synonyms:
Basic fibroblast growth factor | FGF-2 | FGF2 | FGF2_HUMAN | FGFB | Fibroblast growth factor 2 (bFGF) | Fibroblast growth factor receptor 2 (FGF-2) | HBGF-2 | Heparin-binding growth factor 2
Type:
Protein
Mol. Mass.:
30803.89
Organism:
Homo sapiens (Human)
Description:
P09038
Residue:
288
Sequence:
MVGVGGGDVEDVTPRPGGCQISGRGARGCNGIPGAAAWEAALPRRRPRRHPSVNPRSRAAGSPRTRGRRTEERPSGSRLGDRGRGRALPGGRLGGRGRGRAPERVGGRGRGRGTAAPRAAPAARGSRPGPAGTMAAGSITTLPALPEDGGSGAFPPGHFKDPKRLYCKNGGFFLRIHPDGRVDGVREKSDPHIKLQLQAEERGVVSIKGVCANRYLAMKEDGRLLASKCVTDECFFFERLESNNYNTYRSRKYTSWYVALKRTGQYKLGSKTGPGQKAILFLPMSAKS