Reaction Details Report a problem with these data
Target
Neuropeptide FF receptor 2
Ligand
BDBM50583766
Substrate
n/a
Meas. Tech.
ChEMBL_2158117 (CHEMBL5042867)
Ki
1450±n/a nM
Citation
Quillet, R; Schneider, S; Utard, V; Drieu la Rochelle, A; Elhabazi, K; Henningsen, JB; Gizzi, P; Schmitt, M; Kugler, V; Simonneaux, V; Ilien, B; Simonin, F; Bihel, F Identification of an J Med Chem 64:7555-7564 (2021) [PubMed] Article
More Info.:
Target
Name:
Neuropeptide FF receptor 2
Synonyms:
G-protein coupled receptor 74 | Gpr74 | NPFF2_MOUSE | Neuropeptide NPFF receptor | Npff2 | Npffr2
Type:
PROTEIN
Mol. Mass.:
47466.10
Organism:
Mus musculus
Description:
ChEMBL_119166
Residue:
417
Sequence:
MSEKWDSNSSESWNHIWSGNDTQHHWYSDINITYVNYYLHQPQVAAVFISSYLLIFVLCMVGNTVVCFIVIRNRHMHTVTNFFILNLAISDLLVGIFCMPITLLDNIIAGWPFGSSMCKISGLVQGISVAASVFTLVAIAVDRFRCVVYPFKPKLTVKTAFVTIVIIWGLAIAIMTPSAIMLHVQEEKYYRVRLSSHNKTSTVYWCREDWPRHEMRRIYTTVLFATIYLAPLSLIVIMYARIGASLFKTAAHCTGKQRPVQWHVSKKKQKVIKMLLTVALLFILSWLPLWTLMMLSDYTDLSPNKLRIINIYIYPFAHWLAFCNSSVNPIIYGFFNENFRNGFQDAFQICQKKAKPQEAYSLRAKRNIVINTSGLLVQEPVSQNPGGENLGCGKSADNPTQESLIEEMGEATNSTVA