Reaction Details Report a problem with these data
Target
Cannabinoid receptor 2
Ligand
BDBM50213614
Substrate
n/a
Meas. Tech.
ChEMBL_2186029 (CHEMBL5098111)
EC50
32±n/a nM
Citation
Navarro, G; Gonzalez, A; Sánchez-Morales, A; Casajuana-Martin, N; Gómez-Ventura, M; Cordomí, A; Busqué, F; Alibés, R; Pardo, L; Franco, R Design of Negative and Positive Allosteric Modulators of the Cannabinoid CB J Med Chem 64:9354-9364 (2021) [PubMed]
More Info.:
Target
Name:
Cannabinoid receptor 2
Synonyms:
CANNABINOID CB2 | CB-2 | CB2 | CB2A | CB2B | CNR2 | CNR2_HUMAN | CX5 | Cannabinoid CB2 receptor | Cannabinoid receptor 2 (CB2) | Cannabinoid receptor 2 (CB2R) | hCB2
Type:
G Protein-Coupled Receptor (GPCR)
Mol. Mass.:
39690.94
Organism:
Human
Description:
P34972
Residue:
360
Sequence:
MEECWVTEIANGSKDGLDSNPMKDYMILSGPQKTAVAVLCTLLGLLSALENVAVLYLILSSHQLRRKPSYLFIGSLAGADFLASVVFACSFVNFHVFHGVDSKAVFLLKIGSVTMTFTASVGSLLLTAIDRYLCLRYPPSYKALLTRGRALVTLGIMWVLSALVSYLPLMGWTCCPRPCSELFPLIPNDYLLSWLLFIAFLFSGIIYTYGHVLWKAHQHVASLSGHQDRQVPGMARMRLDVRLAKTLGLVLAVLLICWFPVLALMAHSLATTLSDQVKKAFAFCSMLCLINSMVNPVIYALRSGEIRSSAHHCLAHWKKCVRGLGSEAKEEAPRSSVTETEADGKITPWPDSRDLDLSDC