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Target
P2Y purinoceptor 14
Ligand
BDBM50209659
Substrate
n/a
Meas. Tech.
ChEMBL_434326 (CHEMBL917907)
EC50
350±n/a nM
Citation
 Ko, H; Fricks, I; Ivanov, AA; Harden, TK; Jacobson, KA Structure-activity relationship of uridine 5'-diphosphoglucose analogues as agonists of the human P2Y14 receptor. J Med Chem 50:2030-9 (2007) [PubMed]  Article 
Target
Name:
P2Y purinoceptor 14
Synonyms:
P2Y14_HUMAN | P2RY14 | GPR105 | KIAA0001 | Purinergic receptor P2Y14 | Insulin Receptor-Related Protein (INSRR)
Type:
PROTEIN
Mol. Mass.:
38991.62
Organism:
Human
Description:
ChEMBL_1502487
Residue:
338
Sequence:
MINSTSTQPPDESCSQNLLITQQIIPVLYCMVFIAGILLNGVSGWIFFYVPSSKSFIIYLKNIVIADFVMSLTFPFKILGDSGLGPWQLNVFVCRVSAVLFYVNMYVSIVFFGLISFDRYYKIVKPLWTSFIQSVSYSKLLSVIVWMLMLLLAVPNIILTNQSVREVTQIKCIELKSELGRKWHKASNYIFVAIFWIVFLLLIVFYTAITKKIFKSHLKSSRNSTSVKKKSSRNIFSIVFVFFVCFVPYHIARIPYTKSQTEAHYSCQSKEILRYMKEFTLLLSAANVCLDPIIYFFLCQPFREILCKKLHIPLKAQNDLDISRIKRGNTTLESTDTL
  
Inhibitor
Name:
BDBM50209659
Synonyms:
uridine 5'-[3-alpha-D-glucopyranosyl dihydrogen diphosphate] | UDP-alpha-D-glucose
Type:
Small organic molecule
Emp. Form.:
TBD
Mol. Mass.:
TBD
SMILES:
TBD
Structure:
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