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Target
Cytochrome c oxidase subunit NDUFA4
Ligand
BDBM50652792
Substrate
n/a
Meas. Tech.
ChEMBL_2515062
Kd
13491±n/a nM
Citation
 Tröster, A; Heinzlmeir, S; Berger, BT; Gande, SL; Saxena, K; Sreeramulu, S; Linhard, V; Nasiri, AH; Bolte, M; Müller, S; Kuster, B; Médard, G; Kudlinzki, D; Schwalbe, H NVP-BHG712: Effects of Regioisomers on the Affinity and Selectivity toward the EPHrin Family. ChemMedChem 13:1629-1633[PubMed] 
Target
Name:
Cytochrome c oxidase subunit NDUFA4
Synonyms:
NDUA4_HUMAN | NDUFA4 | NADH-ubiquinone oxidoreductase MLRQ subunit
Type:
PROTEIN
Mol. Mass.:
9374.28
Organism:
Human
Description:
ChEMBL_321338
Residue:
81
Sequence:
MLRQIIGQAKKHPSLIPLFVFIGTGATGATLYLLRLALFNPDVCWDRNNPEPWNKLGPNDQYKFYSVNVDYSKLKKERPDF
  
Inhibitor
Name:
BDBM50652792
Synonyms:
CHEMBL3752910
Type:
Small organic molecule
Emp. Form.:
C26H20F3N7O
Mol. Mass.:
503.49
SMILES:
Cc1ccc(C(=O)Nc2cccc(C(F)(F)F)c2)cc1Nc1nc(-c2cccnc2)nc2c1cnn2C
Structure:
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