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Target
5-hydroxytryptamine receptor 4
Ligand
BDBM50241836
Substrate
n/a
Meas. Tech.
ChEMBL_526859 (CHEMBL979354)
Ki
>10000±n/a nM
Citation
 Hedner, E; Sjögren, M; Frändberg, PA; Johansson, T; Göransson, U; Dahlström, M; Jonsson, P; Nyberg, F; Bohlin, L Brominated cyclodipeptides from the marine sponge Geodia barretti as selective 5-HT ligands. J Nat Prod 69:1421-4 (2006) [PubMed]  Article 
Target
Name:
5-hydroxytryptamine receptor 4
Synonyms:
Serotonin Receptor 4 | 5-HT-4 | 5-HT4S | 5-HT4 | Serotonin (5-HT3) receptor | 5-HT4d | 5-hydroxytryptamine receptor 4 | 5-HT4hb | 5-HT4a | Serotonin (5-HT) receptor | Serotonin 4 (5-HT4) receptor | 5-HT4b | 5-HT4c | 5HT4R_HUMAN | HTR4 | 5-hydroxytryptamine receptor 4 (5-HT4)
Type:
Enzyme
Mol. Mass.:
43767.54
Organism:
Human
Description:
Q13639
Residue:
388
Sequence:
MDKLDANVSSEEGFGSVEKVVLLTFLSTVILMAILGNLLVMVAVCWDRQLRKIKTNYFIVSLAFADLLVSVLVMPFGAIELVQDIWIYGEVFCLVRTSLDVLLTTASIFHLCCISLDRYYAICCQPLVYRNKMTPLRIALMLGGCWVIPTFISFLPIMQGWNNIGIIDLIEKRKFNQNSNSTYCVFMVNKPYAITCSVVAFYIPFLLMVLAYYRIYVTAKEHAHQIQMLQRAGASSESRPQSADQHSTHRMRTETKAAKTLCIIMGCFCLCWAPFFVTNIVDPFIDYTVPGQVWTAFLWLGYINSGLNPFLYAFLNKSFRRAFLIILCCDDERYRRPSILGQTVPCSTTTINGSTHVLRDAVECGGQWESQCHPPATSPLVAAQPSDT
  
Inhibitor
Name:
BDBM50241836
Synonyms:
cyclo[(6-bromotryptophan)arginine] | CHEMBL511609
Type:
Small organic molecule
Emp. Form.:
TBD
Mol. Mass.:
TBD
SMILES:
TBD
Structure:
Search PDB for entries with ligand similarity: