Reaction Details Report a problem with these data
Target
5-hydroxytryptamine receptor 1A
Ligand
BDBM50234920
Substrate
n/a
Meas. Tech.
ChEMBL_526854 (CHEMBL979349)
Ki
>10000±n/a nM
Citation
 Hedner, E; Sjögren, M; Frändberg, PA; Johansson, T; Göransson, U; Dahlström, M; Jonsson, P; Nyberg, F; Bohlin, L Brominated cyclodipeptides from the marine sponge Geodia barretti as selective 5-HT ligands. J Nat Prod 69:1421-4 (2006) [PubMed]  Article 
Target
Name:
5-hydroxytryptamine receptor 1A
Synonyms:
5HT1A_HUMAN | ADRB2RL1 | 5-hydroxytryptamine receptor 1A (5-HT-1A) | ADRBRL1 | G-21 | 5-HT-1A | 5-HT1A | HTR1A | Serotonin receptor 1A | Dopamine D2 receptor and serotonin 1a receptor
Type:
n/a
Mol. Mass.:
46122.49
Organism:
Human
Description:
n/a
Residue:
422
Sequence:
MDVLSPGQGNNTTSPPAPFETGGNTTGISDVTVSYQVITSLLLGTLIFCAVLGNACVVAAIALERSLQNVANYLIGSLAVTDLMVSVLVLPMAALYQVLNKWTLGQVTCDLFIALDVLCCTSSILHLCAIALDRYWAITDPIDYVNKRTPRRAAALISLTWLIGFLISIPPMLGWRTPEDRSDPDACTISKDHGYTIYSTFGAFYIPLLLMLVLYGRIFRAARFRIRKTVKKVEKTGADTRHGASPAPQPKKSVNGESGSRNWRLGVESKAGGALCANGAVRQGDDGAALEVIEVHRVGNSKEHLPLPSEAGPTPCAPASFERKNERNAEAKRKMALARERKTVKTLGIIMGTFILCWLPFFIVALVLPFCESSCHMPTLLGAIINWLGYSNSLLNPVIYAYFNKDFQNAFKKIIKCKFCRQ
  
Inhibitor
Name:
BDBM50234920
Synonyms:
Barettin | cyclo[(6-bromo-8-entryptophan)arginine] | (cyclo[(6-bromo-8-entryptophan)arginine]) | CHEMBL255898
Type:
Small organic molecule
Emp. Form.:
TBD
Mol. Mass.:
TBD
SMILES:
TBD
Structure:
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