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Target
Trace amine-associated receptor 1
Ligand
BDBM35929
Substrate
n/a
Meas. Tech.
ChEMBL_489239 (CHEMBL989986)
EC50
3400±n/a nM
Citation
 Lewin, AH; Navarro, HA; Mascarella, SW Structure-activity correlations for beta-phenethylamines at human trace amine receptor 1. Bioorg Med Chem 16:7415-23 (2008) [PubMed]  Article 
Target
Name:
Trace amine-associated receptor 1
Synonyms:
TAAR1_HUMAN | TAAR1 | TA1 | TAR1 | TRAR1 | trace amine-associated receptor 1
Type:
PROTEIN
Mol. Mass.:
39107.47
Organism:
Human
Description:
ChEMBL_792734
Residue:
339
Sequence:
MMPFCHNIINISCVKNNWSNDVRASLYSLMVLIILTTLVGNLIVIVSISHFKQLHTPTNWLIHSMATVDFLLGCLVMPYSMVRSAEHCWYFGEVFCKIHTSTDIMLSSASIFHLSFISIDRYYAVCDPLRYKAKMNILVICVMIFISWSVPAVFAFGMIFLELNFKGAEEIYYKHVHCRGGCSVFFSKISGVLTFMTSFYIPGSIMLCVYYRIYLIAKEQARLISDANQKLQIGLEMKNGISQSKERKAVKTLGIVMGVFLICWCPFFICTVMDPFLHYIIPPTLNDVLIWFGYLNSTFNPMVYAFFYPWFRKALKMMLFGKIFQKDSSRCKLFLELSS
  
Inhibitor
Name:
BDBM35929
Synonyms:
2,2-diphenylethylamine | CHEMBL10780 | 2,2-diphenylethanamine | 2,2-Diphenyl-ethylamine | diphenylalkylamine (DPA), 4a | EN300-13160
Type:
Small organic molecule
Emp. Form.:
TBD
Mol. Mass.:
TBD
SMILES:
TBD
Structure:
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