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Target
Cannabinoid receptor 2
Ligand
BDBM50246588
Substrate
n/a
Meas. Tech.
ChEMBL_558043 (CHEMBL955751)
Ki
749.8±n/a nM
Citation
 Yao, F; Li, C; Vadivel, SK; Bowman, AL; Makriyannis, A Development of novel tail-modified anandamide analogs. Bioorg Med Chem Lett 18:5912-5 (2008) [PubMed]  Article 
Target
Name:
Cannabinoid receptor 2
Synonyms:
CANNABINOID CB2 | CB-2 | CB2 | CNR2_MOUSE | Cannabinoid CB2 receptor | Cannabinoid receptor | Cannabinoid receptor 2 | Cnr2 | mCB2
Type:
Enzyme Catalytic Domain
Mol. Mass.:
38220.43
Organism:
MOUSE
Description:
P47936
Residue:
347
Sequence:
MEGCRETEVTNGSNGGLEFNPMKEYMILSSGQQIAVAVLCTLMGLLSALENMAVLYIILSSRRLRRKPSYLFISSLAGADFLASVIFACNFVIFHVFHGVDSNAIFLLKIGSVTMTFTASVGSLLLTAVDRYLCLCYPPTYKALVTRGRALVALCVMWVLSALISYLPLMGWTCCPSPCSELFPLIPNDYLLGWLLFIAILFSGIIYTYGYVLWKAHRHVATLAEHQDRQVPGIARMRLDVRLAKTLGLVLAVLLICWFPALALMGHSLVTTLSDQVKEAFAFCSMLCLVNSMVNPIIYALRSGEIRSAAQHCLIGWKKYLQGLGPEGKEEGPRSSVTETEADVKTT
  
Inhibitor
Name:
BDBM50246588
Synonyms:
(R,5Z,8Z,11Z,14Z)-19-(furan-2-yl)-N-(1-hydroxypropan-2-yl)nonadeca-5,8,11,14-tetraenamide | CHEMBL516663
Type:
Small organic molecule
Emp. Form.:
C26H39NO3
Mol. Mass.:
413.5928
SMILES:
C[C@H](CO)NC(=O)CCC\C=C/C\C=C/C\C=C/C\C=C/CCCCc1ccco1 |r|
Structure:
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