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Target
Prostaglandin F2-alpha receptor
Ligand
BDBM50350366
Substrate
n/a
Meas. Tech.
ChEMBL_761108 (CHEMBL1815362)
Ki
1400±n/a nM
Citation
 Iwahashi, M; Shimabukuro, A; Onoda, T; Matsunaga, Y; Okada, Y; Matsumoto, R; Nambu, F; Nakai, H; Toda, M Discovery of selective indole-based prostaglandin D2 receptor antagonist. Bioorg Med Chem 19:4574-88 (2011) [PubMed]  Article 
Target
Name:
Prostaglandin F2-alpha receptor
Synonyms:
ProstaglandinF2Alpha | PF2R_MOUSE | Ptgfr
Type:
Enzyme Catalytic Domain
Mol. Mass.:
40714.02
Organism:
Mouse
Description:
ProstaglandinF2Alpha PTGFR MOUSE::P43117
Residue:
366
Sequence:
MSMNSSKQPVSPAAGLIANTTCQTENRLSVFFSIIFMTVGILSNSLAIAILMKAYQRFRQKSKASFLLLASGLVITDFFGHLINGGIAVFVYASDKDWIRFDQSNILCSIFGISMVFSGLCPLFLGSAMAIERCIGVTNPIFHSTKITSKHVKMILSGVCMFAVFVAVLPILGHRDYQIQASRTWCFYNTEHIEDWEDRFYLLFFSFLGLLALGVSFSCNAVTGVTLLRVKFRSQQHRQGRSHHLEMIIQLLAIMCVSCVCWSPFLVTMANIAINGNNSPVTCETTLFALRMATWNQILDPWVYILLRKAVLRNLYKLASRCCGVNIISLHIWELSSIKNSLKVAAISESPAAEKESQQASSEAGL
  
Inhibitor
Name:
BDBM50350366
Synonyms:
CHEMBL1813287
Type:
Small organic molecule
Emp. Form.:
TBD
Mol. Mass.:
TBD
SMILES:
TBD
Structure:
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