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Target
D(1A) dopamine receptor
Ligand
BDBM50088755
Substrate
n/a
Meas. Tech.
ChEBML_59008
Ki
0.700000±n/a nM
Citation
 Tamagnan, G; Baldwin, RM; Kula, NS; Baldessarini, RJ; Innis, RB Cyclopentadienyltricarbonylrheniumbenzazepines: synthesis and binding affinity. Bioorg Med Chem Lett 10:1113-5 (2000) [PubMed]  Article 
Target
Name:
D(1A) dopamine receptor
Synonyms:
DOPAMINE D1 | DRD1_RAT | Dopamine D1 high | Dopamine D1 low | Dopamine receptor | Dopamine receptor D1 | Dopamine1-like | Drd1 | Drd1a
Type:
Enzyme Catalytic Domain
Mol. Mass.:
49429.75
Organism:
RAT
Description:
P18901
Residue:
446
Sequence:
MAPNTSTMDEAGLPAERDFSFRILTACFLSLLILSTLLGNTLVCAAVIRFRHLRSKVTNFFVISLAVSDLLVAVLVMPWKAVAEIAGFWPLGPFCNIWVAFDIMCSTASILNLCVISVDRYWAISSPFQYERKMTPKAAFILISVAWTLSVLISFIPVQLSWHKAKPTWPLDGNFTSLEDTEDDNCDTRLSRTYAISSSLISFYIPVAIMIVTYTSIYRIAQKQIRRISALERAAVHAKNCQTTAGNGNPVECAQSESSFKMSFKRETKVLKTLSVIMGVFVCCWLPFFISNCMVPFCGSEETQPFCIDSITFDVFVWFGWANSSLNPIIYAFNADFQKAFSTLLGCYRLCPTTNNAIETVSINNNGAVVFSSHHEPRGSISKDCNLVYLIPHAVGSSEDLKKEEAGGIAKPLEKLSPALSVILDYDTDVSLEKIQPVTHSGQHST
  
Inhibitor
Name:
BDBM50088755
Synonyms:
5-(2-Bromo-phenyl)-8-chloro-3-methyl-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-ol | CHEMBL13325 | SCH-23390
Type:
Small organic molecule
Emp. Form.:
C17H17BrClNO
Mol. Mass.:
366.68
SMILES:
CN1CCc2cc(Cl)c(O)cc2C(C1)c1ccccc1Br
Structure:
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