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Target
Vasopressin V2 receptor
Ligand
BDBM35667
Substrate
n/a
Meas. Tech.
ChEMBL_215172 (CHEMBL821345)
Kd
1.5±n/a nM
Citation
 Pavo, I; Slaninova, J; Klein, U; Fahrenholz, F Enhanced selectivity of oxytocin antagonists containing sarcosine in position 7. J Med Chem 37:255-9 (1994) [PubMed]  Article 
Target
Name:
Vasopressin V2 receptor
Synonyms:
VASOPRESSIN V2 | V2R_BOVIN | AVPR2 | Vasopressin V2 receptor
Type:
Enzyme Catalytic Domain
Mol. Mass.:
40248.83
Organism:
Bovine
Description:
VASOPRESSIN V2 AVPR2 BOVINE::P48044
Residue:
370
Sequence:
MFMASTTSAVPWHLSQPTPAGNGSEGELLTARDPLLAQAELALLSTVFVAVALSNGLVLGALVRRGRRGRWAPMHVFIGHLCLADLAVALFQVLPQLAWDATDRFRGPDALCRAVKYLQMVGMYASSYMILAMTLDRHRAICRPMLAHRHGGGTHWNRPVLLAWAFSLLFSLPQLFIFAQRDVDGSGVLDCWARFAEPWGLRAYVTWIALMVFVAPALGIAACQVLIFREIHASLGPGPVPRAGGPRRGCRPGSPAEGARVSAAVAKTVKMTLVIVIVYVLCWAPFFLVQLWAAWDPEAPREGPPFVLLMLLASLNSCTNPWIYASFSSSISSELRSLLCCTWRRAPPSPGPQEESCATASSFLAKDTPS
  
Inhibitor
Name:
BDBM35667
Synonyms:
[3H]Argipressin tannate | AVP | [3H]Arginine vasopressin | CHEMBL373742 | [3H]vasopressin | US10131692, 44 (AVP)
Type:
radiolabeled ligand
Emp. Form.:
TBD
Mol. Mass.:
TBD
SMILES:
TBD
Structure:
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