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Target
5-hydroxytryptamine receptor 1D
Ligand
BDBM50056947
Substrate
n/a
Meas. Tech.
ChEMBL_1956 (CHEMBL617563)
Ki
6920±n/a nM
Citation
el Ahmad, Y; Laurent, E; Maillet, P; Talab, A; Teste, JF; Dokhan, R; Tran, G; Ollivier, R New benzocycloalkylpiperazines, potent and selective 5-HT1A receptor ligands. J Med Chem 40:952-60 (1997) [PubMed] Article
More Info.:
Target
Name:
5-hydroxytryptamine receptor 1D
Synonyms:
5HT1D_PIG | HTR1D | Serotonin 1d (5-HT1d) receptor
Type:
PROTEIN
Mol. Mass.:
32680.56
Organism:
Sus scrofa
Description:
ChEMBL_1963
Residue:
291
Sequence:
AMTDLLVSILVMPISIPYTITQTWSFGQLLCDIWLSSDITCCTASILHLCVIALDRYWAITDALEYSKRRTAGHAAAMIAIVWAISICISIPPLFWRQARAHEEISDCLVNTSQISYTIYSTCGAFYIPSLLLIILYGRIYRAARNRILNPPSLYGKRFTTAHLITGSAGSSLCSLNPSLHEGHSHSAGSPLFFNHVKIKLADSVLERKRISAARERKATKTLGIILGAFIICWLPFFVASLVLPICRDSCWIHPALFDFFTWLGYLNSLINPIIYTVFNEEFRQAFQKVV