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Target
P2Y purinoceptor 1
Ligand
BDBM50076474
Substrate
n/a
Meas. Tech.
ChEMBL_147720 (CHEMBL759190)
EC50
2990±n/a nM
Citation
 Nandanan, E; Jang, SY; Moro, S; Kim, HO; Siddiqui, MA; Russ, P; Marquez, VE; Busson, R; Herdewijn, P; Harden, TK; Boyer, JL; Jacobson, KA Synthesis, biological activity, and molecular modeling of ribose-modified deoxyadenosine bisphosphate analogues as P2Y(1) receptor ligands. J Med Chem 43:829-42 (2000) [PubMed]  Article 
Target
Name:
P2Y purinoceptor 1
Synonyms:
P2RY1_MELGA | P2RY1
Type:
n/a
Mol. Mass.:
41199.64
Organism:
Wild turkey
Description:
n/a
Residue:
362
Sequence:
MTEALISAALNGTQPELLAGGWAAGNASTKCSLTKTGFQFYYLPTVYILVFITGFLGNSVAIWMFVFHMRPWSGISVYMFNLALADFLYVLTLPALIFYYFNKTDWIFGDVMCKLQRFIFHVNLYGSILFLTCISVHRYTGVVHPLKSLGRLKKKNAVYVSSLVWALVVAVIAPILFYSGTGVRRNKTITCYDTTADEYLRSYFVYSMCTTVFMFCIPFIVILGCYGLIVKALIYKDLDNSPLRRKSIYLVIIVLTVFAVSYLPFHVMKTLNLRARLDFQTPQMCAFNDKVYATYQVTRGLASLNSCVDPILYFLAGDTFRRRLSRATRKSSRRSEPNVQSKSEEMTLNILTEYKQNGDTSL
  
Inhibitor
Name:
BDBM50076474
Synonyms:
Phosphoric acid mono-[5-(6-amino-purin-9-yl)-2-phosphonooxymethyl-tetrahydro-pyran-3-yl] ester | CHEMBL416252
Type:
Small organic molecule
Emp. Form.:
n/a
Mol. Mass.:
n/a
SMILES:
Nc1ncnc2n(cnc12)C1COC(COP(O)(O)=O)C(C1)OP(O)(O)=O
Structure:
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