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Target
Mu-type opioid receptor
Ligand
BDBM50375296
Substrate
n/a
Meas. Tech.
ChEMBL_470717 (CHEMBL934558)
IC50
129.1±n/a nM
Citation
 Salvadori, S; Fiorini, S; Trapella, C; Porreca, F; Davis, P; Sasaki, Y; Ambo, A; Marczak, ED; Lazarus, LH; Balboni, G Role of benzimidazole (Bid) in the delta-opioid agonist pseudopeptide H-Dmt-Tic-NH-CH(2)-Bid (UFP-502). Bioorg Med Chem 16:3032-8 (2008) [PubMed]  Article 
Target
Name:
Mu-type opioid receptor
Synonyms:
M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO
Type:
Enzyme Catalytic Domain
Mol. Mass.:
11165.58
Organism:
GUINEA PIG
Description:
P97266
Residue:
98
Sequence:
YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSIFTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
  
Inhibitor
Name:
BDBM50375296
Synonyms:
CHEMBL258704
Type:
Small organic molecule
Emp. Form.:
C29H30N4O3S
Mol. Mass.:
514.639
SMILES:
Cc1cc(O)cc(C)c1C[C@H](N)C(=O)N1Cc2ccccc2C[C@H]1C(=O)NCc1nc2ccccc2s1
Structure:
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