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Target
Transcriptional activator protein TraR
Ligand
BDBM50350708
Substrate
n/a
Meas. Tech.
ChEMBL_762769 (CHEMBL1816071)
IC50
10000±n/a nM
Citation
 McInnis, CE; Blackwell, HE Thiolactone modulators of quorum sensing revealed through library design and screening. Bioorg Med Chem 19:4820-8 (2011) [PubMed]  Article 
Target
Name:
Transcriptional activator protein TraR
Synonyms:
TRAR_RHIRD | traR
Type:
PROTEIN
Mol. Mass.:
26741.83
Organism:
Rhizobium radiobacter
Description:
ChEMBL_765233
Residue:
234
Sequence:
MQHWLDKLTDLAAIEGDECILKTGLADIADHFGFTGYAYLHIQHRHITAVTNYHRQWQSTYFDKKFEALDPVVKRARSRKHIFTWSGEHERPTLSKDERAFYDHASDFGIRSGITIPIKTANGFMSMFTMASDKPVIDLDREIDAVAAAATIGQIHARISFLRTTPTAEDAAWLDPKEATYLRWIAVGKTMEEIADVEGVKYNSVRVKLREAMKRFDVRSKAHLTALAIRRKLI
  
Inhibitor
Name:
BDBM50350708
Synonyms:
CHEMBL1814832
Type:
Small organic molecule
Emp. Form.:
C11H19NO2S
Mol. Mass.:
229.339
SMILES:
CCCCCCC(=O)N[C@H]1CCSC1=O |r|
Structure:
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