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Target
Ubiquitin carboxyl-terminal hydrolase 5
Ligand
BDBM50437693
Substrate
n/a
Meas. Tech.
ChEMBL_974343 (CHEMBL2411922)
Ki
12500±n/a nM
Citation
Okada, K; Ye, YQ; Taniguchi, K; Yoshida, A; Akiyama, T; Yoshioka, Y; Onose, J; Koshino, H; Takahashi, S; Yajima, A; Abe, N; Yajima, S Vialinin A is a ubiquitin-specific peptidase inhibitor. Bioorg Med Chem Lett 23:4328-31 (2013) [PubMed] Article
More Info.:
Target
Name:
Ubiquitin carboxyl-terminal hydrolase 5
Synonyms:
Deubiquitinating enzyme 5 | ISOT | Isopeptidase T | UBP5_HUMAN | USP5 | Ubiquitin thioesterase 5 | Ubiquitin-specific-processing protease 5
Type:
PROTEIN
Mol. Mass.:
95751.44
Organism:
Homo sapiens (Human)
Description:
ChEMBL_974329
Residue:
858
Sequence:
MAELSEEALLSVLPTIRVPKAGDRVHKDECAFSFDTPESEGGLYICMNTFLGFGKQYVERHFNKTGQRVYLHLRRTRRPKEEDPATGTGDPPRKKPTRLAIGVEGGFDLSEEKFELDEDVKIVILPDYLEIARDGLGGLPDIVRDRVTSAVEALLSADSASRKQEVQAWDGEVRQVSKHAFSLKQLDNPARIPPCGWKCSKCDMRENLWLNLTDGSILCGRRYFDGSGGNNHAVEHYRETGYPLAVKLGTITPDGADVYSYDEDDMVLDPSLAEHLSHFGIDMLKMQKTDKTMTELEIDMNQRIGEWELIQESGVPLKPLFGPGYTGIRNLGNSCYLNSVVQVLFSIPDFQRKYVDKLEKIFQNAPTDPTQDFSTQVAKLGHGLLSGEYSKPVPESGDGERVPEQKEVQDGIAPRMFKALIGKGHPEFSTNRQQDAQEFFLHLINMVERNCRSSENPNEVFRFLVEEKIKCLATEKVKYTQRVDYIMQLPVPMDAALNKEELLEYEEKKRQAEEEKMALPELVRAQVPFSSCLEAYGAPEQVDDFWSTALQAKSVAVKTTRFASFPDYLVIQIKKFTFGLDWVPKKLDVSIEMPEELDISQLRGTGLQPGEEELPDIAPPLVTPDEPKGSLGFYGNEDEDSFCSPHFSSPTSPMLDESVIIQLVEMGFPMDACRKAVYYTGNSGAEAAMNWVMSHMDDPDFANPLILPGSSGPGSTSAAADPPPEDCVTTIVSMGFSRDQALKALRATNNSLERAVDWIFSHIDDLDAEAAMDISEGRSAADSISESVPVGPKVRDGPGKYQLFAFISHMGTSTMCGHYVCHIKKEGRWVIYNDQKVCASEKPPKDLGYIYFYQRVAS