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Target
Delta-type opioid receptor
Ligand
BDBM50114372
Substrate
n/a
Meas. Tech.
ChEMBL_1511478 (CHEMBL3606827)
Ki
0.340000±n/a nM
Citation
Loriga, G; Lazzari, P; Manca, I; Ruiu, S; Falzoi, M; Murineddu, G; Bottazzi, ME; Pinna, G; Pinna, GA Novel diazabicycloalkane delta opioid agonists. Bioorg Med Chem 23:5527-38 (2015) [PubMed] Article
More Info.:
Target
Name:
Delta-type opioid receptor
Synonyms:
DOR-1 | K56 | MSL-2 | OPIATE Delta | OPRD_MOUSE | Opioid receptors; mu and delta | Oprd1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
40577.25
Organism:
MOUSE
Description:
P32300
Residue:
372
Sequence:
MELVPSARAELQSSPLVNLSDAFPSAFPSAGANASGSPGARSASSLALAIAITALYSAVCAVGLLGNVLVMFGIVRYTKLKTATNIYIFNLALADALATSTLPFQSAKYLMETWPFGELLCKAVLSIDYYNMFTSIFTLTMMSVDRYIAVCHPVKALDFRTPAKAKLINICIWVLASGVGVPIMVMAVTQPRDGAVVCMLQFPSPSWYWDTVTKICVFLFAFVVPILIITVCYGLMLLRLRSVRLLSGSKEKDRSLRRITRMVLVVVGAFVVCWAPIHIFVIVWTLVDINRRDPLVVAALHLCIALGYANSSLNPVLYAFLDENFKRCFRQLCRTPCGRQEPGSLRRPRQATTRERVTACTPSDGPGGGAAA