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Target
5-hydroxytryptamine receptor 4
Ligand
BDBM50056415
Substrate
n/a
Ki
3.98±n/a nM
Comments
PDSP_1620
Citation
 Hegde, SS; Eglen, RM Peripheral 5-HT4 receptors. FASEB J 10:1398-407 (1996) [PubMed]  Article 
Target
Name:
5-hydroxytryptamine receptor 4
Synonyms:
5-HT4 | 5-hydroxytryptamine receptor 4 | 5HT4R_CAVPO | HTR4 | Serotonin 4 (5-HT4) receptor
Type:
Enzyme Catalytic Domain
Mol. Mass.:
43735.29
Organism:
GUINEA PIG
Description:
5-HT4 HTR4 GUINEA PIG::O70528
Residue:
388
Sequence:
MDKLDANVSSKEGFGSVEKVVLLTFLSAVILMAILGNLLVMVAVCRDRQLRKIKTNYFIVSLAFADLLVSVLVMPFGAIELVQDIWVYGEMFCLVRTSLDVLLTTASIFHLCCISLDRYYAICCQPLVYRNKMTPLRIALMLGGCWVIPMFISFLPIMQGWNNIGIVDLIEKRKFNQNSNSTYCVFMVNKPYAITCSVVAFYIPFLLMVLAYYRIYVTAKEHARQIQVLQRAGAPAEGRPQPADQHSTHRMRTETKAAKTLCIIMGCFCLCWAPFFVTNIVDPFIDYTVPGQLWTAFLWLGYINSGLNPFLYAFLNKSFRRAFLIILCCDDERYRRPSILGQTVPCSTTTINGSTHVLRDTVECGGQWESQCHPAASSPLVAAQPIDT
  
Inhibitor
Name:
BDBM50056415
Synonyms:
2-piperidinopropyl 4-amino-5-chloro-2-methoxybenzoate | 4-Amino-5-chloro-2-methoxy-benzoic acid 3-piperidin-1-yl-propyl ester | CHEMBL83954 | RS 23597 | RS-23597-190
Type:
Small organic molecule
Emp. Form.:
C16H23ClN2O3
Mol. Mass.:
326.818
SMILES:
COc1cc(N)c(Cl)cc1C(=O)OCCCN1CCCCC1
Structure:
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