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Target
5-hydroxytryptamine receptor 1B
Ligand
BDBM81790
Substrate
n/a
Ki
>10000±n/a nM
Comments
PDSP_287
Citation
 Schoemaker, H; Claustre, Y; Fage, D; Rouquier, L; Chergui, K; Curet, O; Oblin, A; Gonon, F; Carter, C; Benavides, J; Scatton, B Neurochemical characteristics of amisulpride, an atypical dopamine D2/D3 receptor antagonist with both presynaptic and limbic selectivity. J Pharmacol Exp Ther 280:83-97 (1997) [PubMed] 
Target
Name:
5-hydroxytryptamine receptor 1B
Synonyms:
5-HT1B | Serotonin 1 (5-HT1) receptor | Serotonin receptor 1B | 5-HT-1B | 5-hydroxytryptamine receptor 1B (5HT1B) | 5HT1B_RAT | Htr1b | 5ht1b | Serotonin 1B/1D receptor
Type:
Protein
Mol. Mass.:
43173.33
Organism:
Rat
Description:
P28564
Residue:
386
Sequence:
MEEQGIQCAPPPPATSQTGVPLANLSHNCSADDYIYQDSIALPWKVLLVALLALITLATTLSNAFVIATVYRTRKLHTPANYLIASLAVTDLLVSILVMPISTMYTVTGRWTLGQVVCDFWLSSDITCCTASIMHLCVIALDRYWAITDAVDYSAKRTPKRAAIMIVLVWVFSISISLPPFFWRQAKAEEEVLDCFVNTDHVLYTVYSTVGAFYLPTLLLIALYGRIYVEARSRILKQTPNKTGKRLTRAQLITDSPGSTSSVTSINSRVPEVPSESGSPVYVNQVKVRVSDALLEKKKLMAARERKATKTLGIILGAFIVCWLPFFIISLVMPICKDACWFHMAIFDFFNWLGYLNSLINPIIYTMSNEDFKQAFHKLIRFKCTG
  
Inhibitor
Name:
BDBM81790
Synonyms:
NSC_2159 | CAS_71675-85-9 | Amisulpride | US10167256, Amisulpride | US10259786, Amisulpride
Type:
Small organic molecule
Emp. Form.:
TBD
Mol. Mass.:
TBD
SMILES:
TBD
Structure:
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