Reaction Details Report a problem with these data
Target
D(3) dopamine receptor
Ligand
BDBM81790
Substrate
n/a
Ki
2.9±n/a nM
Comments
PDSP_287
Citation
Schoemaker, H; Claustre, Y; Fage, D; Rouquier, L; Chergui, K; Curet, O; Oblin, A; Gonon, F; Carter, C; Benavides, J; Scatton, B Neurochemical characteristics of amisulpride, an atypical dopamine D2/D3 receptor antagonist with both presynaptic and limbic selectivity. J Pharmacol Exp Ther 280:83-97 (1997) [PubMed]
More Info.:
Target
Name:
D(3) dopamine receptor
Synonyms:
DOPAMINE D3 | DRD3
Type:
Enzyme Catalytic Domain
Mol. Mass.:
40792.06
Organism:
BOVINE
Description:
F1N454
Residue:
367
Sequence:
MAPLNQLGGHINATCAAENSTGAGRARPHAYYALSYCALILAIVFGNVLVCVAVLKERALQTTTNYLVVSLAVADLLVATLVMPWVVYLEVTGGVWNFSRVCCDVFVTLDVMMCTASILNLCAISIDRYTAVVMPVHYQQGTGQSSCRRVALMITAVWLLSFAVSCPLLFGFNTTGDPSICSISNPDFVLYSSVVSFYLPFGVTVLVYARIYVVLRQRRRKRILTRQNSQCLSVRPSFPQQPLSPGQTHMELKRYYSICQDTALGTPGFQEGEGDLKREGRTRNSLMPLREKKATQMLVIVLGTFIVCWLPFFLTHVLNTHCRACHVSPQLYSATTWLGYVNSALNPVIYTTFNIEFRKAFLKILSC