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Target
D(3) dopamine receptor
Ligand
BDBM21398
Substrate
n/a
Ki
6.5±n/a nM
Comments
PDSP_918
Citation
 Schoemaker, H; Claustre, Y; Fage, D; Rouquier, L; Chergui, K; Curet, O; Oblin, A; Gonon, F; Carter, C; Benavides, J; Scatton, B Neurochemical characteristics of amisulpride, an atypical dopamine D2/D3 receptor antagonist with both presynaptic and limbic selectivity. J Pharmacol Exp Ther 280:83-97 (1997) [PubMed] 
Target
Name:
D(3) dopamine receptor
Synonyms:
DOPAMINE D3 | DRD3
Type:
Enzyme Catalytic Domain
Mol. Mass.:
40792.06
Organism:
Bovine
Description:
F1N454
Residue:
367
Sequence:
MAPLNQLGGHINATCAAENSTGAGRARPHAYYALSYCALILAIVFGNVLVCVAVLKERALQTTTNYLVVSLAVADLLVATLVMPWVVYLEVTGGVWNFSRVCCDVFVTLDVMMCTASILNLCAISIDRYTAVVMPVHYQQGTGQSSCRRVALMITAVWLLSFAVSCPLLFGFNTTGDPSICSISNPDFVLYSSVVSFYLPFGVTVLVYARIYVVLRQRRRKRILTRQNSQCLSVRPSFPQQPLSPGQTHMELKRYYSICQDTALGTPGFQEGEGDLKREGRTRNSLMPLREKKATQMLVIVLGTFIVCWLPFFLTHVLNTHCRACHVSPQLYSATTWLGYVNSALNPVIYTTFNIEFRKAFLKILSC
  
Inhibitor
Name:
BDBM21398
Synonyms:
4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1-(4-fluoro-phenyl)-butan-1-one;propionate(HCl) | Haloperidol, 1 | CHEMBL545608 | CHEMBL54 | 4-[4-(4-chlorophenyl)-4-hydroxypiperidin-1-yl]-1-(4-fluorophenyl)butan-1-one | Haloperidol | US20240317745, Compound haloperidol
Type:
Small organic molecule
Emp. Form.:
TBD
Mol. Mass.:
TBD
SMILES:
TBD
Structure:
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