Target
Galanin receptor type 1
Ligand
BDBM50307254
Substrate
n/a
Ki
0.9±n/a nM
Comments
PDSP_1162
Citation
 Howard, ADTan, CShiao, LLPalyha, OCMcKee, KKWeinberg, DHFeighner, SDCascieri, MASmith, RGVan Der Ploeg, LHSullivan, KA Molecular cloning and characterization of a new receptor for galanin. FEBS Lett 405:285-90 (1997) [PubMed]  Article 
Target
Name:
Galanin receptor type 1
Synonyms:
Galanin receptor type 1 | Galanin R1 | GALR1_RAT | Galr1 | Galnr | Galnr1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
38883.91
Organism:
Rat
Description:
Galanin R1 GALR1 RAT::Q62805
Residue:
346
Sequence:
MELAPVNLSEGNGSDPEPPAEPRPLFGIGVENFITLVVFGLIFAMGVLGNSLVITVLARSKPGKPRSTTNLFILNLSIADLAYLLFCIPFQATVYALPTWVLGAFICKFIHYFFTVSMLVSIFTLAAMSVDRYVAIVHSRRSSSLRVSRNALLGVGFIWALSIAMASPVAYYQRLFHRDSNQTFCWEHWPNQLHKKAYVVCTFVFGYLLPLLLICFCYAKVLNHLHKKLKNMSKKSEASKKKTAQTVLVVVVVFGISWLPHHVIHLWAEFGAFPLTPASFFFRITAHCLAYSNSSVNPIIYAFLSENFRKAYKQVFKCRVCNESPHGDAKEKNRIDTPPSTNCTHV
  
Inhibitor
Name:
BDBM50307254
Synonyms:
M40 | CHEMBL604990 | GWTLNSAGYLLGPPPALALA-CONH2
Type:
Small organic molecule
Emp. Form.:
TBD
Mol. Mass.:
TBD
SMILES:
TBD
Structure:
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