Target
Galanin receptor type 2
Ligand
BDBM50273370
Substrate
n/a
Ki
0.43±n/a nM
Comments
PDSP_3167
Citation
 Howard, ADTan, CShiao, LLPalyha, OCMcKee, KKWeinberg, DHFeighner, SDCascieri, MASmith, RGVan Der Ploeg, LHSullivan, KA Molecular cloning and characterization of a new receptor for galanin. FEBS Lett 405:285-90 (1997) [PubMed]  Article 
Target
Name:
Galanin receptor type 2
Synonyms:
Galanin R2 | Galanin receptor type 2 | GALR2_RAT | Galr2 | Galnr2 | Galanin receptor 2
Type:
Enzyme Catalytic Domain
Mol. Mass.:
40697.04
Organism:
Rat
Description:
Galanin R2 GALR2 RAT::O08726
Residue:
372
Sequence:
MNGSGSQGAENTSQEGGSGGWQPEAVLVPLFFALIFLVGTVGNALVLAVLLRGGQAVSTTNLFILNLGVADLCFILCCVPFQATIYTLDDWVFGSLLCKAVHFLIFLTMHASSFTLAAVSLDRYLAIRYPLHSRELRTPRNALAAIGLIWGLALLFSGPYLSYYRQSQLANLTVCHPAWSAPRRRAMDLCTFVFSYLLPVLVLSLTYARTLRYLWRTVDPVTAGSGSQRAKRKVTRMIIIVAVLFCLCWMPHHALILCVWFGRFPLTRATYALRILSHLVSYANSCVNPIVYALVSKHFRKGFRKICAGLLRPAPRRASGRVSILAPGNHSGSMLEQESTDLTQVSEAAGPLVPPPALPNCTASSRTLDPAC
  
Inhibitor
Name:
BDBM50273370
Synonyms:
CHEMBL503473 | M35 | Galanin (1-13)-bradikinin(2-9) | Galanin-(1-13)-bradykinin-(2-9)-amide | GWTLNSAGYLLGPPPGFSPFR-CONH2
Type:
Small organic molecule
Emp. Form.:
TBD
Mol. Mass.:
TBD
SMILES:
TBD
Structure:
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