Reaction Details Report a problem with these data
Target
VIP peptides
Ligand
BDBM85078
Substrate
n/a
Ki
3.4±n/a nM
Comments
PDSP_1607
Citation
 Xia, M; Sreedharan, SP; Bolin, DR; Gaufo, GO; Goetzl, EJ Novel cyclic peptide agonist of high potency and selectivity for the type II vasoactive intestinal peptide receptor. J Pharmacol Exp Ther 281:629-33 (1997) [PubMed] 
Target
Name:
VIP peptides
Synonyms:
VIP_HUMAN | VIP
Type:
Enzyme Catalytic Domain
Mol. Mass.:
19168.43
Organism:
Human
Description:
P01282
Residue:
170
Sequence:
MDTRNKAQLLVLLTLLSVLFSQTSAWPLYRAPSALRLGDRIPFEGANEPDQVSLKEDIDMLQNALAENDTPYYDVSRNARHADGVFTSDFSKLLGQLSAKKYLESLMGKRVSSNISEDPVPVKRHSDAVFTDNYTRLRKQMAVKKYLNSILNGKRSSEGESPDFPEELEK
  
Inhibitor
Name:
BDBM85078
Synonyms:
CAS_150828-75-4 | Ro 25-1392
Type:
Small organic molecule
Emp. Form.:
n/a
Mol. Mass.:
1309.85
SMILES:
CCCCCCCCC[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H]1CC(=O)NCCCC[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](C)NC(=O)C(C)C)C(=O)N[C@@H](Cc2ccccc2)C(=O)N[C@@H](C(C)CC)C(=O)NC(CC(N)=O)C(=O)N1)C(C)CC)C(N)=O |r|
Structure:
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