Reaction Details Report a problem with these data
Target
Galanin receptor type 2
Ligand
BDBM50307254
Substrate
n/a
Ki
2.88±n/a nM
Comments
PDSP_1162
Citation
 Wang, S; He, C; Hashemi, T; Bayne, M Cloning and expressional characterization of a novel galanin receptor. Identification of different pharmacophores within galanin for the three galanin receptor subtypes. J Biol Chem 272:31949-52 (1997) [PubMed]  Article 
Target
Name:
Galanin receptor type 2
Synonyms:
Galanin R2 | Galanin receptor type 2 | GALR2_RAT | Galr2 | Galnr2 | Galanin receptor 2
Type:
Enzyme Catalytic Domain
Mol. Mass.:
40697.04
Organism:
Rat
Description:
Galanin R2 GALR2 RAT::O08726
Residue:
372
Sequence:
MNGSGSQGAENTSQEGGSGGWQPEAVLVPLFFALIFLVGTVGNALVLAVLLRGGQAVSTTNLFILNLGVADLCFILCCVPFQATIYTLDDWVFGSLLCKAVHFLIFLTMHASSFTLAAVSLDRYLAIRYPLHSRELRTPRNALAAIGLIWGLALLFSGPYLSYYRQSQLANLTVCHPAWSAPRRRAMDLCTFVFSYLLPVLVLSLTYARTLRYLWRTVDPVTAGSGSQRAKRKVTRMIIIVAVLFCLCWMPHHALILCVWFGRFPLTRATYALRILSHLVSYANSCVNPIVYALVSKHFRKGFRKICAGLLRPAPRRASGRVSILAPGNHSGSMLEQESTDLTQVSEAAGPLVPPPALPNCTASSRTLDPAC
  
Inhibitor
Name:
BDBM50307254
Synonyms:
M40 | CHEMBL604990 | GWTLNSAGYLLGPPPALALA-CONH2
Type:
Small organic molecule
Emp. Form.:
TBD
Mol. Mass.:
TBD
SMILES:
TBD
Structure:
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