Reaction Details Report a problem with these data
Target
Galanin receptor type 3
Ligand
BDBM50273370
Substrate
n/a
Ki
7.5±n/a nM
Comments
PDSP_851
Citation
 Wang, S; He, C; Hashemi, T; Bayne, M Cloning and expressional characterization of a novel galanin receptor. Identification of different pharmacophores within galanin for the three galanin receptor subtypes. J Biol Chem 272:31949-52 (1997) [PubMed]  Article 
Target
Name:
Galanin receptor type 3
Synonyms:
Galanin R3 | Galanin receptor type 3 | GALR3_RAT | Galr3 | Galnr3
Type:
Enzyme Catalytic Domain
Mol. Mass.:
40439.51
Organism:
Rat
Description:
Galanin R3 GALR3 RAT::O88626
Residue:
370
Sequence:
MADIQNISLDSPGSVGAVAVPVIFALIFLLGMVGNGLVLAVLLQPGPSAWQEPRSTTDLFILNLAVADLCFILCCVPFQAAIYTLDAWLFGAFVCKTVHLLIYLTMYASSFTLAAVSLDRYLAVRHPLRSRALRTPRNARAAVGLVWLLAALFSAPYLSYYGTVRYGALELCVPAWEDARRRALDVATFAAGYLLPVAVVSLAYGRTLCFLWAAVGPAGAAAAEARRRATGRAGRAMLAVAALYALCWGPHHALILCFWYGRFAFSPATYACRLASHCLAYANSCLNPLVYSLASRHFRARFRRLWPCGRRRHRHHHRAHRALRRVQPASSGPAGYPGDARPRGWSMEPRGDALRGGGETRLTLSPRGPQ
  
Inhibitor
Name:
BDBM50273370
Synonyms:
CHEMBL503473 | M35 | Galanin (1-13)-bradikinin(2-9) | Galanin-(1-13)-bradykinin-(2-9)-amide | GWTLNSAGYLLGPPPGFSPFR-CONH2
Type:
Small organic molecule
Emp. Form.:
TBD
Mol. Mass.:
TBD
SMILES:
TBD
Structure:
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