Reaction Details Report a problem with these data
Target
Galanin receptor type 1
Ligand
BDBM85169
Substrate
n/a
Ki
407.38±n/a nM
Comments
PDSP_3183
Citation
 Smith, KE; Walker, MW; Artymyshyn, R; Bard, J; Borowsky, B; Tamm, JA; Yao, WJ; Vaysse, PJ; Branchek, TA; Gerald, C; Jones, KA Cloned human and rat galanin GALR3 receptors. Pharmacology and activation of G-protein inwardly rectifying K+ channels. J Biol Chem 273:23321-6 (1998) [PubMed]  Article 
Target
Name:
Galanin receptor type 1
Synonyms:
Galanin receptor type 1 | Galanin R1 | GALR1_RAT | Galr1 | Galnr | Galnr1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
38883.91
Organism:
Rat
Description:
Galanin R1 GALR1 RAT::Q62805
Residue:
346
Sequence:
MELAPVNLSEGNGSDPEPPAEPRPLFGIGVENFITLVVFGLIFAMGVLGNSLVITVLARSKPGKPRSTTNLFILNLSIADLAYLLFCIPFQATVYALPTWVLGAFICKFIHYFFTVSMLVSIFTLAAMSVDRYVAIVHSRRSSSLRVSRNALLGVGFIWALSIAMASPVAYYQRLFHRDSNQTFCWEHWPNQLHKKAYVVCTFVFGYLLPLLLICFCYAKVLNHLHKKLKNMSKKSEASKKKTAQTVLVVVVVFGISWLPHHVIHLWAEFGAFPLTPASFFFRITAHCLAYSNSSVNPIIYAFLSENFRKAYKQVFKCRVCNESPHGDAKEKNRIDTPPSTNCTHV
  
Inhibitor
Name:
BDBM85169
Synonyms:
Galanin [D-Trp2], porcine | Galanin (1-29), porcine
Type:
Small organic molecule
Emp. Form.:
TBD
Mol. Mass.:
TBD
SMILES:
TBD
Structure:
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