Target
Galanin receptor type 1
Ligand
BDBM85072
Substrate
n/a
Ki
0.60±n/a nM
Comments
PDSP_864
Citation
 Smith, KEWalker, MWArtymyshyn, RBard, JBorowsky, BTamm, JAYao, WJVaysse, PJBranchek, TAGerald, CJones, KA Cloned human and rat galanin GALR3 receptors. Pharmacology and activation of G-protein inwardly rectifying K+ channels. J Biol Chem 273:23321-6 (1998) [PubMed]  Article 
Target
Name:
Galanin receptor type 1
Synonyms:
Galanin receptor type 1 | Galanin R1 | GALR1_RAT | Galr1 | Galnr | Galnr1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
38883.91
Organism:
Rat
Description:
Galanin R1 GALR1 RAT::Q62805
Residue:
346
Sequence:
MELAPVNLSEGNGSDPEPPAEPRPLFGIGVENFITLVVFGLIFAMGVLGNSLVITVLARSKPGKPRSTTNLFILNLSIADLAYLLFCIPFQATVYALPTWVLGAFICKFIHYFFTVSMLVSIFTLAAMSVDRYVAIVHSRRSSSLRVSRNALLGVGFIWALSIAMASPVAYYQRLFHRDSNQTFCWEHWPNQLHKKAYVVCTFVFGYLLPLLLICFCYAKVLNHLHKKLKNMSKKSEASKKKTAQTVLVVVVVFGISWLPHHVIHLWAEFGAFPLTPASFFFRITAHCLAYSNSSVNPIIYAFLSENFRKAYKQVFKCRVCNESPHGDAKEKNRIDTPPSTNCTHV
  
Inhibitor
Name:
BDBM85072
Synonyms:
Galanin, Human
Type:
Small organic molecule
Emp. Form.:
TBD
Mol. Mass.:
TBD
SMILES:
TBD
Structure:
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