Reaction Details Report a problem with these data
Target
Galanin receptor type 1
Ligand
BDBM85073
Substrate
n/a
Ki
0.65±n/a nM
Comments
PDSP_3166
Citation
Smith, KE; Walker, MW; Artymyshyn, R; Bard, J; Borowsky, B; Tamm, JA; Yao, WJ; Vaysse, PJ; Branchek, TA; Gerald, C; Jones, KA Cloned human and rat galanin GALR3 receptors. Pharmacology and activation of G-protein inwardly rectifying K+ channels. J Biol Chem 273:23321-6 (1998) [PubMed] Article
More Info.:
Target
Name:
Galanin receptor type 1
Synonyms:
GALR1_RAT | Galanin R1 | Galanin receptor type 1 | Galnr | Galnr1 | Galr1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
38883.91
Organism:
RAT
Description:
Galanin R1 GALR1 RAT::Q62805
Residue:
346
Sequence:
MELAPVNLSEGNGSDPEPPAEPRPLFGIGVENFITLVVFGLIFAMGVLGNSLVITVLARSKPGKPRSTTNLFILNLSIADLAYLLFCIPFQATVYALPTWVLGAFICKFIHYFFTVSMLVSIFTLAAMSVDRYVAIVHSRRSSSLRVSRNALLGVGFIWALSIAMASPVAYYQRLFHRDSNQTFCWEHWPNQLHKKAYVVCTFVFGYLLPLLLICFCYAKVLNHLHKKLKNMSKKSEASKKKTAQTVLVVVVVFGISWLPHHVIHLWAEFGAFPLTPASFFFRITAHCLAYSNSSVNPIIYAFLSENFRKAYKQVFKCRVCNESPHGDAKEKNRIDTPPSTNCTHV