Reaction Details Report a problem with these data
Target
Galanin receptor type 3
Ligand
BDBM50307254
Substrate
n/a
Ki
79.43±n/a nM
Comments
PDSP_1162
Citation
 Smith, KE; Walker, MW; Artymyshyn, R; Bard, J; Borowsky, B; Tamm, JA; Yao, WJ; Vaysse, PJ; Branchek, TA; Gerald, C; Jones, KA Cloned human and rat galanin GALR3 receptors. Pharmacology and activation of G-protein inwardly rectifying K+ channels. J Biol Chem 273:23321-6 (1998) [PubMed]  Article 
Target
Name:
Galanin receptor type 3
Synonyms:
Galanin R3 | Galanin receptor type 3 | GALR3_RAT | Galr3 | Galnr3
Type:
Enzyme Catalytic Domain
Mol. Mass.:
40439.51
Organism:
Rat
Description:
Galanin R3 GALR3 RAT::O88626
Residue:
370
Sequence:
MADIQNISLDSPGSVGAVAVPVIFALIFLLGMVGNGLVLAVLLQPGPSAWQEPRSTTDLFILNLAVADLCFILCCVPFQAAIYTLDAWLFGAFVCKTVHLLIYLTMYASSFTLAAVSLDRYLAVRHPLRSRALRTPRNARAAVGLVWLLAALFSAPYLSYYGTVRYGALELCVPAWEDARRRALDVATFAAGYLLPVAVVSLAYGRTLCFLWAAVGPAGAAAAEARRRATGRAGRAMLAVAALYALCWGPHHALILCFWYGRFAFSPATYACRLASHCLAYANSCLNPLVYSLASRHFRARFRRLWPCGRRRHRHHHRAHRALRRVQPASSGPAGYPGDARPRGWSMEPRGDALRGGGETRLTLSPRGPQ
  
Inhibitor
Name:
BDBM50307254
Synonyms:
M40 | CHEMBL604990 | GWTLNSAGYLLGPPPALALA-CONH2
Type:
Small organic molecule
Emp. Form.:
TBD
Mol. Mass.:
TBD
SMILES:
TBD
Structure:
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