Reaction Details Report a problem with these data
Target
Muscarinic acetylcholine receptor M4
Ligand
BDBM81799
Substrate
n/a
Ki
32.35±n/a nM
Comments
PDSP_931
Citation
 Chelala, JL; Kilani, A; Miller, MJ; Martin, RJ; Ernsberger, P Muscarinic receptor binding sites of the M4 subtype in porcine lung parenchyma. Pharmacol Toxicol 83:200-7 (1998) [PubMed]  Article 
Target
Name:
Muscarinic acetylcholine receptor M4
Synonyms:
CHRM4 | CHRM4 protein | Cholinergic, muscarinic M4
Type:
Enzyme Catalytic Domain
Mol. Mass.:
30028.84
Organism:
bovine
Description:
A6QQE4
Residue:
271
Sequence:
MTVLYVHISLASRSRVHKHRPEGPKEKKAKTLAFLKSPLMKQSVKKPPPPGDTTARGELRNGKLEEAPPPVLPPPPRPMADKDTSNESSSGSATQNTKERPPTELSTTEATTPATPAPPLQPRTLNPASKWSKIQIVTKQTGNECVTAIEIVPATPAGMRPAANVARKFASIARSQVRKKRQMAARERKVTRTIFAILLAFILTWTPYNVMVLVNTFCQSCIPETVWSIGYWLCYVNSTINPACYALCNATFKKTFRHLLLCQYRNIGTAR
  
Inhibitor
Name:
BDBM81799
Synonyms:
CAS_98299-40-2 | HHSiD | NSC_3602 | hexahydrosiladifenidol
Type:
Small organic molecule
Emp. Form.:
C20H33NOSi
Mol. Mass.:
331.5676
SMILES:
O[Si](CCCN1CCCCC1)(C1CCCCC1)c1ccccc1
Structure:
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