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Target
Galanin receptor type 1
Ligand
BDBM50307254
Substrate
n/a
Ki
2.40±n/a nM
Comments
PDSP_1162
Citation
 Borowsky, B; Walker, MW; Huang, LY; Jones, KA; Smith, KE; Bard, J; Branchek, TA; Gerald, C Cloning and characterization of the human galanin GALR2 receptor. Peptides 19:1771-81 (1998) [PubMed]  Article 
Target
Name:
Galanin receptor type 1
Synonyms:
Galanin receptor 1 | Galanin receptor type 1 | GAL1-R | Galanin R1 | GALR1_HUMAN | GALR1 | GALNR | GALNR1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
38976.60
Organism:
Human
Description:
Galanin R1 GALR1 HUMAN::P47211
Residue:
349
Sequence:
MELAVGNLSEGNASWPEPPAPEPGPLFGIGVENFVTLVVFGLIFALGVLGNSLVITVLARSKPGKPRSTTNLFILNLSIADLAYLLFCIPFQATVYALPTWVLGAFICKFIHYFFTVSMLVSIFTLAAMSVDRYVAIVHSRRSSSLRVSRNALLGVGCIWALSIAMASPVAYHQGLFHPRASNQTFCWEQWPDPRHKKAYVVCTFVFGYLLPLLLICFCYAKVLNHLHKKLKNMSKKSEASKKKTAQTVLVVVVVFGISWLPHHIIHLWAEFGVFPLTPASFLFRITAHCLAYSNSSVNPIIYAFLSENFRKAYKQVFKCHIRKDSHLSDTKESKSRIDTPPSTNCTHV
  
Inhibitor
Name:
BDBM50307254
Synonyms:
M40 | CHEMBL604990 | GWTLNSAGYLLGPPPALALA-CONH2
Type:
Small organic molecule
Emp. Form.:
TBD
Mol. Mass.:
TBD
SMILES:
TBD
Structure:
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