Reaction Details Report a problem with these data
Target
Cysteinyl leukotriene receptor 1
Ligand
BDBM85673
Substrate
n/a
Ki
2.3±n/a nM
Comments
PDSP_1248
Citation
 Nothacker, HP; Wang, Z; Zhu, Y; Reinscheid, RK; Lin, SH; Civelli, O Molecular cloning and characterization of a second human cysteinyl leukotriene receptor: discovery of a subtype selective agonist. Mol Pharmacol 58:1601-8 (2000) [PubMed]  Article 
Target
Name:
Cysteinyl leukotriene receptor 1
Synonyms:
Leukotriene Cysteinyl 1 | Cysteinyl leukotriene receptor | HMTMF81 | LTD4 receptor | Cysteinyl leukotriene D4 receptor | HG55 | CLTR1_HUMAN | CYSLTR1 | CYSLT1 | Cysteinyl leukotriene receptor 1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
38565.16
Organism:
Human
Description:
Leukotriene Cysteinyl 1 CYSLTR1 HUMAN::Q9Y271
Residue:
337
Sequence:
MDETGNLTVSSATCHDTIDDFRNQVYSTLYSMISVVGFFGNGFVLYVLIKTYHKKSAFQVYMINLAVADLLCVCTLPLRVVYYVHKGIWLFGDFLCRLSTYALYVNLYCSIFFMTAMSFFRCIAIVFPVQNINLVTQKKARFVCVGIWIFVILTSSPFLMAKPQKDEKNNTKCFEPPQDNQTKNHVLVLHYVSLFVGFIIPFVIIIVCYTMIILTLLKKSMKKNLSSHKKAIGMIMVVTAAFLVSFMPYHIQRTIHLHFLHNETKPCDSVLRMQKSVVITLSLAASNCCFDPLLYFFSGGNFRKRLSTFRKHSLSSVTYVPRKKASLPEKGEEICKV
  
Inhibitor
Name:
BDBM85673
Synonyms:
NSC_5311297 | CAS_5311297 | Montelukast
Type:
Small organic molecule
Emp. Form.:
TBD
Mol. Mass.:
TBD
SMILES:
TBD
Structure:
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