Reaction Details Report a problem with these data
Target
Alpha-2B adrenergic receptor
Ligand
BDBM81773
Substrate
n/a
Ki
95.3±n/a nM
Comments
PDSP_340
Citation
Naselsky, DP; Ashton, D; Ruffolo, RR; Hieble, JP Rabbit alpha2-adrenoceptors: both platelets and adipocytes have alpha2A-pharmacology. J Pharmacol Exp Ther 298:219-25 (2001) [PubMed]
More Info.:
Target
Name:
Alpha-2B adrenergic receptor
Synonyms:
ADA2B_RABIT | ADRA2B | Alpha-2B adrenergic receptor | adrenergic Alpha2
Type:
Enzyme Catalytic Domain
Mol. Mass.:
42909.14
Organism:
RABBIT
Description:
adrenergic Alpha2 0 RABBIT::O77830
Residue:
394
Sequence:
AIAAVITFLILFTIFGNALVILAVLTSRSLRAPQNLFLVSLAAADILVATLIIPFSLANELLGYWYFRRTWCEVYLALDVLFCTSSIVHLCAISLDRYWAVSRALEYNCKRTPRRIKCIILTVWLIAAAISLPPLIYKGDQGPQPHGAPQCKLNQEAWYILSSSLGSFFVPCLIMILVYLRIYLIAKRSHRRGPRAKGGPGEGESRQACPVPGGPSASAKLPTLATPVASASEANGPSKPAGEKEEGETPEDPGTQALPPGWATLPNSGQGQKEGVSGASLEEEAEEEEEEEEEEDEPQAVPVSPASVGSPPLQQPQGSRVLATLRGQVLVGRGVGAMSGQWWRRRAQLSREKRFTFVLAVVIGVFVLCWFPFFFSYSLSAICPQQCRVPHGLF