Target
Neuropeptide Y receptor type 5
Ligand
BDBM84998
Substrate
n/a
Ki
0.31±n/a nM
Comments
PDSP_1372
Citation
 Holmberg, SKMikko, SBoswell, TZoorob, RLarhammar, D Pharmacological characterization of cloned chicken neuropeptide Y receptors Y1 and Y5. J Neurochem 81:462-71 (2002) [PubMed]  Article 
Target
Name:
Neuropeptide Y receptor type 5
Synonyms:
NPY-Y5 | NPY5R
Type:
Enzyme Catalytic Domain
Mol. Mass.:
50065.15
Organism:
Chicken
Description:
Q8QFM2
Residue:
443
Sequence:
MDLGFKDYTNRTPTKNTSATTKNFSAWEDYKSSVDDIQYFLIGLYTLISLAGFVGNLLVLTALTKRKQKTIINILIGNLAFSDILVVLFCSPFTLTSVLLDRWMFGTVMCHIMPFLQCTSVLVSTLMLISIAAVRYRMVKYPLSSNLTAKHGYFLIVIIWAVGCAICSPLPVFHKIVDLHKTLNLEALENRLLCIESWPSDSYRIAFTISLLLMQYILPLVCLTASHTSVCRSVGSRLSSKEGKFQENEMINLTLHPSKSAGTEAQPSSHTSWSCALVRKHHRRYSKKTSTVMPAILRQQQDADFRDLPETSGTEKSQLSSSSKFIPGVPICFEMKPEENTEIQDMITVSQSIIRIKTRSRRVFCRLTVLILVFGFSWMPLHLFHIVTDFNATLISNRHFKLVYCICHLLGMMSCCLNPILYGFLNNSIKADLMSLIPCCQIL
  
Inhibitor
Name:
BDBM84998
Synonyms:
NPY 3-36, porcine
Type:
Small organic molecule
Emp. Form.:
C195H295N53O57
Mol. Mass.:
4293.7497
SMILES:
n/a
Structure:
Search PDB for entries with ligand similarity: