Reaction Details Report a problem with these data
Target
AP-2 complex subunit sigma
Ligand
BDBM81790
Substrate
n/a
Ki
>10000±n/a nM
Comments
PDSP_287
Citation
Abbas, AI; Hedlund, PB; Huang, XP; Tran, TB; Meltzer, HY; Roth, BL Amisulpride is a potent 5-HT7 antagonist: relevance for antidepressant actions in vivo. Psychopharmacology (Berl) 205:119-28 (2009) [PubMed] Article
More Info.:
Target
Name:
AP-2 complex subunit sigma
Synonyms:
AP-2 complex subunit sigma | AP2S1_RAT | Ap17 | Ap2s1 | Claps2 | Sigma-2
Type:
Enzyme Catalytic Domain
Mol. Mass.:
17016.49
Organism:
RAT
Description:
Sigma-2 0 RAT::P62744
Residue:
142
Sequence:
MIRFILIQNRAGKTRLAKWYMQFDDDEKQKLIEEVHAVVTVRDAKHTNFVEFRNFKIIYRRYAGLYFCICVDVNDNNLAYLEAIHNFVEVLNEYFHNVCELDLVFNFYKVYTVVDEMFLAGEIRETSQTKVLKQLLMLQSLE