Reaction Details Report a problem with these data
Target
Tyrosine-protein kinase CSK
Ligand
BDBM93207
Substrate
n/a
Meas. Tech.
Fluorescence Assay
pH
7.5000±0.0000
Temperature
298.1500±0.0000 K
IC50
8.4±0.2 nM
Citation
 Brigham, JL; Perera, BG; Maly, DJ A Hexylchloride-Based Catch-and-Release System for Chemical Proteomic Applications. ACS Chem Biol 8:691-9 (2013) [PubMed]  Article 
Target
Name:
Tyrosine-protein kinase CSK
Synonyms:
C-SRC kinase | C-src tyrosine kinase | Protein-tyrosine kinase CYL | Tyrosine Kinase CSK | CSK_HUMAN | CSK
Type:
Tyrosine-protein kinase
Mol. Mass.:
50707.30
Organism:
Human
Description:
P41240
Residue:
450
Sequence:
MSAIQAAWPSGTECIAKYNFHGTAEQDLPFCKGDVLTIVAVTKDPNWYKAKNKVGREGIIPANYVQKREGVKAGTKLSLMPWFHGKITREQAERLLYPPETGLFLVRESTNYPGDYTLCVSCDGKVEHYRIMYHASKLSIDEEVYFENLMQLVEHYTSDADGLCTRLIKPKVMEGTVAAQDEFYRSGWALNMKELKLLQTIGKGEFGDVMLGDYRGNKVAVKCIKNDATAQAFLAEASVMTQLRHSNLVQLLGVIVEEKGGLYIVTEYMAKGSLVDYLRSRGRSVLGGDCLLKFSLDVCEAMEYLEGNNFVHRDLAARNVLVSEDNVAKVSDFGLTKEASSTQDTGKLPVKWTAPEALREKKFSTKSDVWSFGILLWEIYSFGRVPYPRIPLKDVVPRVEKGYKMDAPDGCPPAVYEVMKNCWHLDAAMRPSFLQLREQLEHIKTHELHL
  
Inhibitor
Name:
BDBM93207
Synonyms:
Kinase inhibitor, 5
Type:
Small molecule
Emp. Form.:
TBD
Mol. Mass.:
TBD
SMILES:
TBD
Structure:
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