Reaction Details Report a problem with these data
Target
Mu-type opioid receptor
Ligand
BDBM98006
Substrate
n/a
Meas. Tech.
Radioligand Binding Assay
pH
7.4000±0.0000
Ki
330.6±0.0 nM
Citation
 Zhou, X Phenylpropionamide compounds and the use thereof US Patent  US8481743 Publication Date 7/9/2013 
Target
Name:
Mu-type opioid receptor
Synonyms:
M-OR-1 | MOP | MOR-1 | MUOR1 | Mu Opioid Receptor | Mu opiate receptor | OPIATE Mu | hMOP | mu-type opioid receptor isoform MOR-1 | OPRM_HUMAN | OPRM1 | MOR1
Type:
G Protein-Coupled Receptor (GPCR)
Mol. Mass.:
44789.51
Organism:
Human
Description:
P35372
Residue:
400
Sequence:
MDSSAAPTNASNCTDALAYSSCSPAPSPGSWVNLSHLDGNLSDPCGPNRTDLGGRDSLCPPTGSPSMITAITIMALYSIVCVVGLFGNFLVMYVIVRYTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSIFTLCTMSVDRYIAVCHPVKALDFRTPRNAKIINVCNWILSSAIGLPVMFMATTKYRQGSIDCTLTFSHPTWYWENLLKICVFIFAFIMPVLIITVCYGLMILRLKSVRMLSGSKEKDRNLRRITRMVLVVVAVFIVCWTPIHIYVIIKALVTIPETTFQTVSWHFCIALGYTNSCLNPVLYAFLDENFKRCFREFCIPTSSNIEQQNSTRIRQNTRDHPSTANTVDRTNHQLENLEAETAPLP
  
Inhibitor
Name:
BDBM98006
Synonyms:
US8481743, 2
Type:
Small organic molecule
Emp. Form.:
n/a
Mol. Mass.:
n/a
SMILES:
CCC(=O)N(C1CCN(CCC(c2ccccc2)c2ccccc2)CC1)c1ccccc1
Structure:
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