Target

Ligand

Substrate

Meas. Tech.

Glutathione S-transferase Activity Assay

pH

6.5±n/a

Ki

267350±n/a nM

Citation

 Ekinci, D; Cankaya, M; Gül, Ä°; Coban, TA Susceptibility of cord blood antioxidant enzymes glutathione reductase, glutathione peroxidase and glutathione S-transferase to different antibiotics: in vitro approach. J Enzyme Inhib Med Chem 28:824-9 (2013) [PubMed]  Article Copy BDB DOI

More Info.:

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Name:

Microsomal glutathione S-transferase 1

Synonyms:

GST12 | Glutathione S-transferase (GST) | MGST | MGST1 | MGST1_HUMAN

Type:

Enzyme

Mol. Mass.:

17605.01

Organism:

Homo sapiens (Human)

Description:

P10620

Residue:

155

Sequence:

MVDLTQVMDDEVFMAFASYATIILSKMMLMSTATAFYRLTRKVFANPEDCVAFGKGENAKKYLRTDDRVERVRRAHLNDLENIIPFLGIGLLYSLSGPDPSTAILHFRLFVGARIYHTIAYLTPLPQPNRALSFFVGYGVTLSMAYRLLKSKLYL

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Name:

BDBM50390999

Synonyms:

CEFOPERAZONE

Type:

Small organic molecule

Emp. Form.:

C25H27N9O8S2

Mol. Mass.:

645.667

SMILES:

CCN1CCN(C(=O)N[C@@H](C(=O)N[C@H]2[C@H]3SCC(CSc4nnnn4C)=C(N3C2=O)C(O)=O)c2ccc(O)cc2)C(=O)C1=O |c:26|

Structure:

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