Reaction Details Report a problem with these data
Target
Vasopressin V1b receptor
Ligand
BDBM35667
Substrate
n/a
Meas. Tech.
In Vitro V1b Receptor Assay
EC50
5400±n/a nM
Citation
 Wisniewski, K; Schteingart, C; Riviere, P Vasopressin-2 receptor agonists US Patent  US10131692 Publication Date 11/20/2018 
Target
Name:
Vasopressin V1b receptor
Synonyms:
Vasopressin V3 receptor | AVPR V3 | AVPR V1b | Antidiuretic hormone receptor 1b | V1bR | VASOPRESSIN V1B | Vasopressin V3 | AVPR3 | VPR3 | V1BR_HUMAN | AVPR1B | Vasopressin V1b receptor | Vasopressin V1b receptor (V1b)
Type:
Enzyme
Mol. Mass.:
46985.01
Organism:
Human
Description:
P47901
Residue:
424
Sequence:
MDSGPLWDANPTPRGTLSAPNATTPWLGRDEELAKVEIGVLATVLVLATGGNLAVLLTLGQLGRKRSRMHLFVLHLALTDLAVALFQVLPQLLWDITYRFQGPDLLCRAVKYLQVLSMFASTYMLLAMTLDRYLAVCHPLRSLQQPGQSTYLLIAAPWLLAAIFSLPQVFIFSLREVIQGSGVLDCWADFGFPWGPRAYLTWTTLAIFVLPVTMLTACYSLICHEICKNLKVKTQAWRVGGGGWRTWDRPSPSTLAATTRGLPSRVSSINTISRAKIRTVKMTFVIVLAYIACWAPFFSVQMWSVWDKNAPDEDSTNVAFTISMLLGNLNSCCNPWIYMGFNSHLLPRPLRHLACCGGPQPRMRRRLSDGSLSSRHTTLLTRSSCPATLSLSLSLTLSGRPRPEESPRDLELADGEGTAETIIF
  
Inhibitor
Name:
BDBM35667
Synonyms:
[3H]Argipressin tannate | AVP | [3H]Arginine vasopressin | CHEMBL373742 | [3H]vasopressin | US10131692, 44 (AVP)
Type:
radiolabeled ligand
Emp. Form.:
TBD
Mol. Mass.:
TBD
SMILES:
TBD
Structure:
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