Assay Method Information

Assay Name:  ChEMBL_1813295 (CHEMBL4312869)
Description:  Antagonist activity at human PPARgamma expressed in 293H cells assessed as reduction in rosiglitazone-induced transcriptional response preincubated for 30 mins followed by rosiglitazone addition and measured after 16 hrs by reporter gene-based FRET assay
Affinity data for this assay
 

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