Compile Data Set for Download or QSAR
maximum 50k data
Found 45 of affinity data for UniProtKB/TrEMBL: A9XFY4
TargetNicotinic acetylcholine receptor alpha 5 subunit(Musca domestica)
Dow Agrosciences

Curated by ChEMBL
LigandPNGBDBM50488015(CHEMBL2272685)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]imidacloprid from nicotinic acetylcholine receptor in Musca domestica (house fly) head membrane after 1 hr by liquid scintillatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(Musca domestica)
Dow Agrosciences

Curated by ChEMBL
LigandPNGBDBM50212288((2E)-1-[(6-chloropyridin-3-yl)methyl]-N-nitroimida...)
Affinity DataKi:  4.60nMAssay Description:Displacement of [3H]IMI from Musca domestica (house fly) brain nicotinic acetylcholine receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(Musca domestica)
Dow Agrosciences

Curated by ChEMBL
LigandPNGBDBM50488014(CHEMBL2272690)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]imidacloprid from nicotinic acetylcholine receptor in Musca domestica (house fly) head membrane after 1 hr by liquid scintillatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(Musca domestica)
Dow Agrosciences

Curated by ChEMBL
LigandPNGBDBM50488022(CHEMBL2251976)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]imidacloprid from nicotinic acetylcholine receptor in Musca domestica (house fly) head membrane after 1 hr by liquid scintillatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(Musca domestica)
Dow Agrosciences

Curated by ChEMBL
LigandPNGBDBM50487224(CHEMBL2252498)
Affinity DataKi:  30nMAssay Description:Displacement of [3H]IMI from Musca domestica (house fly) brain nicotinic acetylcholine receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(Musca domestica)
Dow Agrosciences

Curated by ChEMBL
LigandPNGBDBM50487219(CHEMBL2252497)
Affinity DataKi:  150nMAssay Description:Displacement of [3H]IMI from Musca domestica (house fly) brain nicotinic acetylcholine receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(Musca domestica)
Dow Agrosciences

Curated by ChEMBL
LigandPNGBDBM50488017(CHEMBL2272689)
Affinity DataKi:  400nMAssay Description:Displacement of [3H]imidacloprid from nicotinic acetylcholine receptor in Musca domestica (house fly) head membrane after 1 hr by liquid scintillatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(Musca domestica)
Dow Agrosciences

Curated by ChEMBL
LigandPNGBDBM50488024(CHEMBL2272695)
Affinity DataKi:  441nMAssay Description:Displacement of [3H]imidacloprid from nicotinic acetylcholine receptor in Musca domestica (house fly) head membrane after 1 hr by liquid scintillatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(Musca domestica)
Dow Agrosciences

Curated by ChEMBL
LigandPNGBDBM50488016(CHEMBL2272684)
Affinity DataKi:  517nMAssay Description:Displacement of [3H]imidacloprid from nicotinic acetylcholine receptor in Musca domestica (house fly) head membrane after 1 hr by liquid scintillatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(Musca domestica)
Dow Agrosciences

Curated by ChEMBL
LigandPNGBDBM50487229(CHEMBL2252496)
Affinity DataKi:  530nMAssay Description:Displacement of [3H]IMI from Musca domestica (house fly) brain nicotinic acetylcholine receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(Musca domestica)
Dow Agrosciences

Curated by ChEMBL
LigandPNGBDBM50488019(CHEMBL2272691)
Affinity DataKi:  593nMAssay Description:Displacement of [3H]imidacloprid from nicotinic acetylcholine receptor in Musca domestica (house fly) head membrane after 1 hr by liquid scintillatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(Musca domestica)
Dow Agrosciences

Curated by ChEMBL
LigandPNGBDBM50487226(CHEMBL2252501)
Affinity DataKi:  800nMAssay Description:Displacement of [3H]IMI from Musca domestica (house fly) brain nicotinic acetylcholine receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(Musca domestica)
Dow Agrosciences

Curated by ChEMBL
LigandPNGBDBM50487222(CHEMBL2252352)
Affinity DataKi:  1.46E+3nMAssay Description:Displacement of [3H]IMI from Musca domestica (house fly) brain nicotinic acetylcholine receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(Musca domestica)
Dow Agrosciences

Curated by ChEMBL
LigandPNGBDBM50488021(CHEMBL2272694)
Affinity DataKi:  1.53E+3nMAssay Description:Displacement of [3H]imidacloprid from nicotinic acetylcholine receptor in Musca domestica (house fly) head membrane after 1 hr by liquid scintillatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(Musca domestica)
Dow Agrosciences

Curated by ChEMBL
LigandPNGBDBM50487231(CHEMBL2252353)
Affinity DataKi:  1.55E+3nMAssay Description:Displacement of [3H]IMI from Musca domestica (house fly) brain nicotinic acetylcholine receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(Musca domestica)
Dow Agrosciences

Curated by ChEMBL
LigandPNGBDBM50488026(CHEMBL2272686)
Affinity DataKi:  1.78E+3nMAssay Description:Displacement of [3H]imidacloprid from nicotinic acetylcholine receptor in Musca domestica (house fly) head membrane after 1 hr by liquid scintillatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(Musca domestica)
Dow Agrosciences

Curated by ChEMBL
LigandPNGBDBM50487227(CHEMBL447459)
Affinity DataKi:  2.27E+3nMAssay Description:Displacement of [3H]IMI from Musca domestica (house fly) brain nicotinic acetylcholine receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(Musca domestica)
Dow Agrosciences

Curated by ChEMBL
LigandPNGBDBM50487225(CHEMBL2252499)
Affinity DataKi:  2.30E+3nMAssay Description:Displacement of [3H]IMI from Musca domestica (house fly) brain nicotinic acetylcholine receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(Musca domestica)
Dow Agrosciences

Curated by ChEMBL
LigandPNGBDBM50487223(CHEMBL2252495)
Affinity DataKi:  2.66E+3nMAssay Description:Displacement of [3H]IMI from Musca domestica (house fly) brain nicotinic acetylcholine receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(Musca domestica)
Dow Agrosciences

Curated by ChEMBL
LigandPNGBDBM50487232(CHEMBL2252503)
Affinity DataKi:  2.77E+3nMAssay Description:Displacement of [3H]IMI from Musca domestica (house fly) brain nicotinic acetylcholine receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(Musca domestica)
Dow Agrosciences

Curated by ChEMBL
LigandPNGBDBM50487220(CHEMBL2252350)
Affinity DataKi:  2.90E+3nMAssay Description:Displacement of [3H]IMI from Musca domestica (house fly) brain nicotinic acetylcholine receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(Musca domestica)
Dow Agrosciences

Curated by ChEMBL
LigandPNGBDBM50488020(CHEMBL2272693)
Affinity DataKi:  3.34E+3nMAssay Description:Displacement of [3H]imidacloprid from nicotinic acetylcholine receptor in Musca domestica (house fly) head membrane after 1 hr by liquid scintillatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(Musca domestica)
Dow Agrosciences

Curated by ChEMBL
LigandPNGBDBM50488018(CHEMBL2272688)
Affinity DataKi:  3.83E+3nMAssay Description:Displacement of [3H]imidacloprid from nicotinic acetylcholine receptor in Musca domestica (house fly) head membrane after 1 hr by liquid scintillatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(Musca domestica)
Dow Agrosciences

Curated by ChEMBL
LigandPNGBDBM50488023(CHEMBL2272692)
Affinity DataKi:  3.92E+3nMAssay Description:Displacement of [3H]imidacloprid from nicotinic acetylcholine receptor in Musca domestica (house fly) head membrane after 1 hr by liquid scintillatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(Musca domestica)
Dow Agrosciences

Curated by ChEMBL
LigandPNGBDBM50487233(CHEMBL2252500)
Affinity DataKi:  5.20E+3nMAssay Description:Displacement of [3H]IMI from Musca domestica (house fly) brain nicotinic acetylcholine receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(Musca domestica)
Dow Agrosciences

Curated by ChEMBL
LigandPNGBDBM50488025(CHEMBL2272687)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]imidacloprid from nicotinic acetylcholine receptor in Musca domestica (house fly) head membrane after 1 hr by liquid scintillatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(Musca domestica)
Dow Agrosciences

Curated by ChEMBL
LigandPNGBDBM50488027(CHEMBL2272683)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]imidacloprid from nicotinic acetylcholine receptor in Musca domestica (house fly) head membrane after 1 hr by liquid scintillatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(Musca domestica)
Dow Agrosciences

Curated by ChEMBL
LigandPNGBDBM50487228(CHEMBL2252504)
Affinity DataKi:  1.60E+4nMAssay Description:Displacement of [3H]IMI from Musca domestica (house fly) brain nicotinic acetylcholine receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(Musca domestica)
Dow Agrosciences

Curated by ChEMBL
LigandPNGBDBM50487230(CHEMBL2252502)
Affinity DataKi:  1.70E+4nMAssay Description:Displacement of [3H]IMI from Musca domestica (house fly) brain nicotinic acetylcholine receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(Musca domestica)
Dow Agrosciences

Curated by ChEMBL
LigandPNGBDBM50487221(CHEMBL2252351)
Affinity DataKi:  2.60E+4nMAssay Description:Displacement of [3H]IMI from Musca domestica (house fly) brain nicotinic acetylcholine receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(Musca domestica)
Dow Agrosciences

Curated by ChEMBL
LigandPNGBDBM50487218(CHEMBL2252349)
Affinity DataKi:  2.60E+4nMAssay Description:Displacement of [3H]IMI from Musca domestica (house fly) brain nicotinic acetylcholine receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(Musca domestica)
Dow Agrosciences

Curated by ChEMBL
LigandPNGBDBM50486231(CHEBI:39177 | CLOTHIANIDINE)
Affinity DataIC50:  1.80nMAssay Description:Displacement of [3H]IMI from nicotinic acetylcholine receptor in Musca domestica (house fly) head membrane after 90 min by filter binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(Musca domestica)
Dow Agrosciences

Curated by ChEMBL
LigandPNGBDBM50212288((2E)-1-[(6-chloropyridin-3-yl)methyl]-N-nitroimida...)
Affinity DataIC50:  2.60nMAssay Description:Displacement of [3H]IMI from nicotinic acetylcholine receptor in Musca domestica (house fly) head membrane after 90 min by filter binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(Musca domestica)
Dow Agrosciences

Curated by ChEMBL
LigandPNGBDBM50487983(CHEMBL148390)
Affinity DataIC50:  7.10nMAssay Description:Displacement of [3H]IMI from nicotinic acetylcholine receptor in Musca domestica (house fly) head membrane after 90 min by filter binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(Musca domestica)
Dow Agrosciences

Curated by ChEMBL
LigandPNGBDBM50487979(IMIDACLOTHIZ)
Affinity DataIC50:  12nMAssay Description:Displacement of [3H]IMI from nicotinic acetylcholine receptor in Musca domestica (house fly) head membrane after 90 min by filter binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(Musca domestica)
Dow Agrosciences

Curated by ChEMBL
LigandPNGBDBM50487985(CHEMBL2269823)
Affinity DataIC50:  14nMAssay Description:Displacement of [3H]IMI from nicotinic acetylcholine receptor in Musca domestica (house fly) head membrane after 90 min by filter binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(Musca domestica)
Dow Agrosciences

Curated by ChEMBL
LigandPNGBDBM50487980(DESMETHYLTHIAMETHOXAM)
Affinity DataIC50:  16nMAssay Description:Displacement of [3H]IMI from nicotinic acetylcholine receptor in Musca domestica (house fly) head membrane after 90 min by filter binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(Musca domestica)
Dow Agrosciences

Curated by ChEMBL
LigandPNGBDBM50212288((2E)-1-[(6-chloropyridin-3-yl)methyl]-N-nitroimida...)
Affinity DataIC50:  20nMAssay Description:Displacement of [3HIMI from nicotinic acetylcholine receptor in Musca domestica (house fly) head membranes incubated for 60 min by liquid scintillati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(Musca domestica)
Dow Agrosciences

Curated by ChEMBL
LigandPNGBDBM50488029((S)-METHYL-IMIDACLOPRID)
Affinity DataIC50:  190nMAssay Description:Displacement of [3HIMI from nicotinic acetylcholine receptor in Musca domestica (house fly) head membranes incubated for 60 min by liquid scintillati...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(Musca domestica)
Dow Agrosciences

Curated by ChEMBL
LigandPNGBDBM50488030((R,S)-METHYL-IMIDACLOPRID)
Affinity DataIC50:  210nMAssay Description:Displacement of [3HIMI from nicotinic acetylcholine receptor in Musca domestica (house fly) head membranes incubated for 60 min by liquid scintillati...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(Musca domestica)
Dow Agrosciences

Curated by ChEMBL
LigandPNGBDBM50488028((R)-METHYL-IMIDACLOPRID)
Affinity DataIC50:  950nMAssay Description:Displacement of [3HIMI from nicotinic acetylcholine receptor in Musca domestica (house fly) head membranes incubated for 60 min by liquid scintillati...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(Musca domestica)
Dow Agrosciences

Curated by ChEMBL
LigandPNGBDBM50143314((+)-Epibatidine | (-)-epibatidine | (1R,2R,4S)-2-(...)
Affinity DataIC50:  1.34E+3nMAssay Description:Displacement of [3HIMI from nicotinic acetylcholine receptor in Musca domestica (house fly) head membranes incubated for 60 min by liquid scintillati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(Musca domestica)
Dow Agrosciences

Curated by ChEMBL
LigandPNGBDBM50143320((+)-epibatidine | (-)-1-epidatidine | (1S,2S,4R)-2...)
Affinity DataIC50:  2.79E+3nMAssay Description:Displacement of [3HIMI from nicotinic acetylcholine receptor in Musca domestica (house fly) head membranes incubated for 60 min by liquid scintillati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(Musca domestica)
Dow Agrosciences

Curated by ChEMBL
LigandPNGBDBM82070(CAS_29790-52-1 | NICOTINE-L (BASE) | Nicotine-D sa...)
Affinity DataIC50:  1.19E+4nMAssay Description:Displacement of [3HIMI from nicotinic acetylcholine receptor in Musca domestica (house fly) head membranes incubated for 60 min by liquid scintillati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(Musca domestica)
Dow Agrosciences

Curated by ChEMBL
LigandPNGBDBM82068(CHEMBL9732 | Nicotine-D salicylate | Nicotine-L sa...)
Affinity DataIC50:  4.22E+5nMAssay Description:Displacement of [3HIMI from nicotinic acetylcholine receptor in Musca domestica (house fly) head membranes incubated for 60 min by liquid scintillati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed